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4-(2-fluorophenoxy)-1-(pyrazine-2-carbonyl)piperidine-4-carboxylic acid
N-methyl-2-oxo-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1-oxaspiro[4.4]nonane-4-carboxamide
3-(azocan-1-yl)-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)propanamide
3-[1-(7-fluoro-3-methyl-1H-indole-2-carbonyl)piperidin-4-yl]phenol
(2S,4S)-4-amino-N-methyl-1-{2-methyl-3-[(pyridin-3-ylmethyl)amino]benzoyl}pyrrolidine-2-carboxamide
1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
1-(piperidin-3-ylmethyl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decane-7-carboxamide
1-(2-benzylphenyl)-3-{[4-(dimethylamino)oxan-4-yl]methyl}urea
1-(cyclopent-1-ene-1-carbonyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
6-(2-aminoethyl)-N,2-dimethyl-N-(quinolin-5-ylmethyl)pyrimidin-4-amine
ethyl 4-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carboxylate
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-{5-[1-(3-chlorophenyl)-1H-pyrrol-2-yl]-4-phenyl-1H-imidazol-1-yl}propane-1,2-diol
(3S,4R)-1-methyl-3-{[methyl(thiophen-3-ylmethyl)amino]methyl}piperidin-4-ol
5-[1-butyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-N-methylpyrimidin-2-amine
2-(ethylamino)-N-[2-(N-methylmethanesulfonamido)ethyl]pyrimidine-5-carboxamide
[(3R,4R)-1-(5-methyl-1,3-benzoxazol-2-yl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4,4-difluoropiperidine
N-cyclopropyl-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine-2-carboxamide
3-(2-oxo-2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,3-oxazolidin-2-one
2-methyl-5-{3-[4-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}pyrazine
dimethyl[(4-methyl-5-{1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
N-(4-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}phenyl)acetamide
3-hydroxy-3-({[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
3-{[(furan-2-ylmethyl)amino]methyl}-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
2-{2-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,2,3,4-tetrahydroisoquinolin-1-yl}acetic acid
N-(1-cycloheptylpiperidin-3-yl)-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2,6-dimethoxyphenyl)-1,2,4-oxadiazole
1-{2-[(dimethyl-1,3-thiazol-4-yl)formamido]ethyl}piperidine-3-carboxamide
3-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-5-phenyl-1,2-oxazole
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-(pyridin-4-yl)-1,4-diazepan-6-ol
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl][(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]methylamine
(1S,5R)-6-(3-ethyl-1H-pyrazole-4-carbonyl)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
2-{[(3S,4S)-3,4-bis(hydroxymethyl)pyrrolidin-1-yl]methyl}-6-methylquinolin-4-ol
3-{2-oxo-2-[2-(2-phenylethyl)morpholin-4-yl]ethyl}-1,2,3-oxadiazol-3-ium-5-olate
4-methoxy-N-(2-methoxyethyl)-2-{[1-(piperidin-4-yl)piperidin-4-yl]oxy}benzamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
3-benzyl-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidine-3-carboxylic acid
N-[4-(3-methoxyphenyl)phenyl]-1-(2-methylpropanoyl)pyrrolidine-2-carboxamide
(3R,4R)-1-(3-methoxy-5-methylthiophene-2-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(3-methylphenoxy)piperidine
9-methyl-3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3,9-diazaspiro[5.6]dodecan-10-one
2-{[(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
4-(5-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(2-hydroxyacetyl)piperidine-4-carboxamide
(3ar,6ar)-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
5-acetyl-N-{1-[(3-chlorophenyl)amino]-2-methylpropan-2-yl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
5-ethyl-N-[(3-methylpyridin-2-yl)methyl]-N-(propan-2-yl)-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2,3,4-trifluorobenzamide