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2-{1-[(4-ethoxyphenyl)methyl]-4-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperazin-2-yl}ethan-1-ol
2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[(2-methoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2,3-dihydro-1-benzofuran-7-carboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
N-cyclopropyl-N-({1-[1-oxo-1-(piperidin-1-yl)propan-2-yl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)[(2-methyl-1H-imidazol-4-yl)methyl](oxolan-2-ylmethyl)amine
1-(cyclopent-1-ene-1-carbonyl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
1-(6-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}pyridin-3-yl)ethan-1-one
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(1H-indol-3-yl)acetamide
(4aR,7aS)-1-{[2,4-bis(prop-2-en-1-yloxy)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(3-methyl-1H-pyrazol-5-yl)methyl]amine
4-(5-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
1-(2-chloro-6-fluoro-3-methylbenzoyl)-3-(3-methoxypropyl)piperidine
2-[2-(dimethylamino)ethyl]-9-(quinoxalin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
7-[(2,3-difluorophenyl)methyl]-2-[(2E)-2-methylbut-2-en-1-yl]-2,7-diazaspiro[4.5]decan-6-one
1,3-dimethyl-5-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)imidazolidine-2,4-dione
(2S)-1-{[4-phenyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}pyrrolidine-2-carboxamide
1-[2-(2-fluorophenoxy)phenyl]-3-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]urea
2-(2-methyl-1,3-thiazol-4-yl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindole-2-carbonyl]-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
1-[2-(cyclopropylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]azetidine
N-[(2-chlorophenyl)methyl]-N-cyclopropyl-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
2-(quinolin-8-yl)pyridin-4-amine
N-[2-(4-methylmorpholin-2-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-3-(1,2-oxazinan-2-yl)propan-1-one
1-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-3-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
4-(1-{[4-(dimethylamino)oxan-4-yl]methyl}-1H-imidazol-2-yl)-2-(prop-2-en-1-yl)phenol
3-(3-chlorophenyl)-6-(2-methylpropyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
6-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-1-phenylpiperazin-2-one
3-({[2-(1H-1,3-benzodiazol-2-yl)ethyl](methyl)amino}methyl)-1,2-dihydroquinolin-2-one
5-(cyclohex-3-ene-1-carbonyl)-N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-4-phenylpyrrolidin-2-one
N-(2-ethoxyphenyl)-3-[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]-3-oxopropanamide
3-{5-[2-(1H-imidazol-2-yl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-pyrazole-5-carboxamide
1,1-dioxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1λ6-thiane-4-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
(1R,5R)-N,N-dimethyl-6-[(5-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-cyclohexaneamido-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(2-methoxyethyl)-N-methyl-1H-1,3-benzodiazole-7-carboxamide
6-hydroxy-N-[3-(2-methoxyphenyl)phenyl]-1,4-oxazepane-4-carboxamide
4-methyl-3-(4-methyl-1H-pyrazol-1-yl)benzamide
(2S,4S)-4-[2-(3-chloro-2,4-difluorophenyl)acetamido]-N-ethyl-1-methylpyrrolidine-2-carboxamide
(3R,4R)-3-cyclopropyl-4-methyl-1-[4-(4-methylpiperazin-1-yl)benzoyl]pyrrolidin-3-ol
N-[(2-chlorophenyl)methyl]-4-oxo-N-(prop-2-en-1-yl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-[2-(3-methoxypyrrolidin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid