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3-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-4,5,6-trimethyl-1,2-dihydropyridin-2-one
3-[3-(2-phenylpyrrolidine-1-carbonyl)phenyl]piperidine
N-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-3-(2,5-dioxoimidazolidin-4-yl)-N-methylpropanamide
3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(2-phenylethyl)piperidine
3-[3-(oxolan-3-yl)-5-{2H,3H-thieno[3,4-b][1,4]dioxin-5-yl}-1H-1,2,4-triazol-1-yl]pyridine
4-(4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)phenol
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-6-methyl-4-oxo-4H-pyran-2-carboxamide
3-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidine-3-carbonyl}pyridine
(3R,5S)-N-(2-methylpropyl)-5-(morpholin-4-ylmethyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
1-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-N-cyclopropylpiperidine-4-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
5-{[3-(3-chlorophenyl)-3-phenylpropanamido]methyl}-N-methylfuran-2-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-ethylpyrimidin-2-amine
2-methyl-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1-(propan-2-yl)piperazine
5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-2-(thiophen-3-yl)pyridine
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}piperidin-2-one
N-[2-(2,5-dimethoxyphenyl)phenyl]propanamide
2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}[(1-methyl-1H-imidazol-2-yl)methyl]amino)ethan-1-ol
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-5-methylpyrazine-2-carboxamide
(4R)-4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-3-methyl-1,3-thiazolidine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(piperidine-1-carbonyl)benzene-1-sulfonamide
2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]-4-(2,5-dimethylthiophen-3-yl)pyrimidine
4-(2-acetylbenzoyl)-1-(3-chlorophenyl)-5-methylpiperazin-2-one
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
2-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-8-fluoro-1,4-dihydroquinolin-4-one
7-cyclopentyl-2-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(cyclopropylmethyl)-8-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
5-[4-(4-ethoxy-3-methylphenyl)butanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
ethyl 4-{1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
1-(oxolan-2-ylmethyl)-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(2,4-difluorophenyl)ethan-1-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
3-{[(2,4-dimethoxyphenyl)methyl]amino}-1-(3-methylpiperidin-1-yl)propan-1-one
N-({7-[2-(2-chloro-4-fluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-sulfonamide
1-[2-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-3-methoxy-1,2-dihydropyridin-2-one
4-[3-(4-propylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]morpholine
3-(1H-indol-5-yl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-3,5-dimethyl-1H-indole-2-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
1-methyl-4-{4-phenyl-5-[5-(1H-pyrazol-5-yl)thiophen-2-yl]-1H-imidazol-1-yl}piperidine
1-cyclobutanecarbonyl-4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]piperidine
4-[(dimethylamino)methyl]-1-(3-phenyl-1,2,4-oxadiazol-5-yl)azepan-4-ol
1-(1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-1-oxopropan-2-yl)pyrrolidin-2-one
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-[4-(pyrrolidin-1-ylmethyl)benzoyl]-1λ6-thiomorpholine-1,1-dione
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(thiophen-2-yl)acetamide
3-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1-[2-(2-methoxyethoxy)phenyl]urea
2-[(2-butylpyrrolidin-1-yl)methyl]benzoic acid
4-(2-fluoro-4,5-dimethoxyphenyl)-7-(2-oxoimidazolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one