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2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
(1S,5R)-6-benzyl-3-[3-(methylsulfanyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-2-(phenylamino)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
6-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}-9H-purin-2-amine
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[3-(morpholin-4-yl)propyl]amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-4-methylpyrimidine-5-carboxamide
8-(4-propylpyrimidine-5-carbonyl)-1-oxa-8-azaspiro[4.5]decane
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(piperidin-4-yl)pyrimidin-2-amine
3-{[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl](methyl)amino}propanamide
3-[2-ethoxy-5-(trifluoromethyl)phenyl]-1-[3-(morpholin-4-yl)propyl]urea
N-methyl-N-(oxolan-2-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N3-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-N5-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
ethyl 2-(1-{5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carbonyl}piperidin-2-yl)acetate
5-methyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-1-propyl-1H-pyrazole-4-carboxamide
6,8-dimethyl-3-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N6-cyclopropyl-N5-methyl-N5-[(5-methylfuran-2-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
4-{5-[3-(dimethylamino)phenyl]-3-methyl-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
2-({[(3R,4R)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(2E)-1-[(4aR,8aS)-6-(2-methoxyacetyl)-decahydro-1,6-naphthyridin-1-yl]-3-(4-fluorophenyl)prop-2-en-1-one
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethyl-1-(2-phenoxyphenyl)urea
N-cyclopentyl-N'-[2-methoxy-1-(pyridin-2-yl)ethyl]-N'-methylbutanediamide
2-[2-(1-tert-butyl-3-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2,3-dihydro-1λ6,2-benzothiazole-1,1,3-trione
N4-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-6-(morpholin-4-yl)pyrimidine-2,4-diamine
2-({[1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
2-methyl-4-(5-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}furan-2-yl)but-3-yn-2-ol
3-[(dimethylamino)methyl]-1-(quinoxaline-5-carbonyl)pyrrolidin-3-ol
(2E)-3-(1H-imidazol-4-yl)-1-{4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}prop-2-en-1-one
N,N-dimethyl-1-[3-({1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)benzoyl]pyrrolidin-3-amine
1-{1-[(2-chlorophenyl)methyl]piperidin-3-yl}-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
1-[cyclohexyl(methyl)amino]-3-[3-(2,3-dihydro-1H-isoindol-2-ylmethyl)phenoxy]propan-2-ol
1-[(3-fluorophenyl)methyl]-4-[3-(pyrrolidin-3-yl)benzoyl]piperazine
(1S,9S)-11-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-N'-(3,5-dimethylphenyl)propanediamide
5-ethyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
4-(4-methylpyrimidin-2-yl)benzamide
(2S,4R)-4-amino-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-(2,4-difluorophenyl)-1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-phenyl-1H-imidazole
2-[2-(4-fluorophenyl)piperidine-1-carbonyl]-6-methoxy-1-methyl-1H-indole
4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperazine-2-carboxylic acid
methyl 2-[({1-[(4-fluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]acetate
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}diethylamine
N-(3,5-dimethoxyphenyl)-2-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]acetamide
2-{4-[(4-methoxyphenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
2-[5-(4-methylpiperazine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1H-1,3-benzodiazole
2-ethoxy-5-[2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-4-yl]benzoic acid
2-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-(3-{[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]amino}propyl)piperidin-4-ol
3-[1-(2-amino-9H-purin-6-yl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{1-[2-(2-methyl-1H-imidazol-1-yl)acetyl]piperidin-3-yl}benzoic acid