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3-{[(3-acetyl-2,4,6-trimethylphenyl)methyl](ethyl)amino}-1λ6-thiolane-1,1-dione
4-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4,6-dimethyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
3-ethyl-5-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-1,2-oxazole-4-carboxamide
(1S,5R)-6-benzyl-3-[(4-methanesulfonylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-1-(piperidin-3-yl)piperidine
1-[cyclohexyl(methyl)amino]-3-[2-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]cyclobutanecarboxamide
1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-N-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4-[7-(2-ethoxypyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
6-methoxy-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[4-methyl-3-(thiophen-2-yl)-1H-pyrazol-1-yl]-N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}acetamide
4-methyl-2-(4H-1,2,4-triazol-4-yl)-5-[3-(trifluoromethyl)phenyl]pyridine
N-[(1-hydroxycyclohexyl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
3-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(4-hydroxypiperidin-1-yl)acetamide
3-phenoxy-N-[1-({[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
2-{5-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4,4,4-trifluorobutan-1-one
1-{1-[(7-hydroxyquinolin-3-yl)methyl]piperidin-4-yl}butan-1-one
2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetic acid
2-butoxy-N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}acetamide
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
7-(2,3-dimethoxyphenyl)-4-[(2,4-dimethylphenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-fluoro-N-{2-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzamide
5-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]quinoxaline
2-{2,7-diazaspiro[4.5]decane-2-carbonyl}-4-methylphenol
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}propanamide
1-[2-({[2-(butan-2-yloxy)-3-methoxyphenyl]methyl}amino)ethyl]imidazolidin-2-one
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[(2-hydroxyethyl)amino]methyl}piperidin-2-one
1-{6-[(3-methoxypropyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}-N,N-dimethylpyrrolidin-3-amine
5-fluoro-4-(morpholin-4-yl)-N-[2-(thiophen-2-yl)ethyl]pyrimidin-2-amine
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-amine
N-{2-[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-N-methylmethanesulfonamide
2-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-N-(2,4-dimethylphenyl)-2-oxoacetamide
4-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N,3,6,7-tetramethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1-benzofuran-2-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-(1-ethyl-1H-pyrazole-5-carbonyl)piperazin-2-one
1-[(2-chlorophenyl)methyl]-N-[1-(pyrimidin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(3-methoxyphenyl)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
1-benzyl-N-[1-(3-methylpyridin-2-yl)propyl]piperidin-4-amine
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-1-(3-methyl-3-phenylpiperidin-1-yl)ethan-1-one
3-[3-(4-methanesulfonylphenyl)phenyl]-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1H-pyrazole
N-[(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]cyclopropanecarboxamide
1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
7-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-5-[2-(piperidin-1-yl)ethyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene