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N-{1-[1-(cyclobutylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
5-(2,4-difluorophenoxymethyl)-N-(oxolan-2-ylmethyl)-N-propyl-1,2-oxazole-3-carboxamide
(1,4-dioxan-2-ylmethyl)({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)methylamine
5-{2-[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-3-(propan-2-yl)-1,2,4-oxadiazole
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(methylsulfanyl)pyrimidin-4-amine
[(2-fluorophenyl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
9-[(2-fluoro-4-methoxyphenyl)methyl]-3-methyl-3,9-diazaspiro[5.6]dodecane
4-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}methyl)-N-(1-methyl-1H-imidazol-2-yl)benzamide
3-methoxy-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}propanamide
N-(3-{7-[(3-methylphenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-3-oxopropyl)acetamide
1-ethyl-4-{5-[5-(hydroxymethyl)furan-2-yl]-4-phenyl-1H-imidazol-1-yl}pyrrolidin-2-one
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-ethyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-cyclohexyl-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
3-[2-(3-aminopyrrolidin-1-yl)-2-oxoethyl]-1-[(2-fluorophenyl)methyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
1-[4-(1H-pyrazol-3-yl)benzoyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-(2,4-difluorophenyl)-1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]propan-1-one
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
2-(ethylamino)-N-[3-(pyridin-4-yl)propyl]pyrimidine-5-carboxamide
8-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
N-[(3R,4R)-1-(3-cyanopyridin-2-yl)-3-hydroxypiperidin-4-yl]-N-ethyl-2,3-difluorobenzamide
3-chloro-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-4-fluoro-1-benzothiophene-2-carboxamide
methyl (1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
3-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
N-methyl-2-propyl-N-(quinoxalin-2-ylmethyl)-1,3-thiazole-4-carboxamide
(1S,5R)-6-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
3-(1,2-oxazinan-2-yl)-N-[4-(pyridin-2-yl)butyl]propanamide
N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)morpholine-2-carboxamide
5-[2-(furan-3-yl)-1H-imidazol-1-yl]-2-(3-methoxyphenoxy)pyridine
6-{[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]amino}pyridine-2-carbonitrile
1-ethyl-N-methyl-N-[1-(pyridin-3-yl)propyl]piperidin-4-amine
methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl})(thiophen-3-ylmethyl)amine
4-{2-[5-(5-methylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyridine
N,3-diethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-4-methyl-1H-pyrazole-5-carboxamide
2-methoxy-N-[1-(2-phenylethyl)-7-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1H-1,3-benzodiazol-5-yl]acetamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropylimidazo[2,1-b][1,3]thiazole-6-carboxamide
(4aR,8aS)-6-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-1-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1-[(3,4-difluorophenyl)methyl]-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
ethyl 4-({[4-(furan-2-yl)phenyl]carbamoyl}amino)piperidine-1-carboxylate
N-(4-fluoro-2-methylphenyl)-4-(2-propoxyethyl)piperazine-1-carboxamide
N-({5-[(5-fluoro-2-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}acetamide
2-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,3-benzodiazole
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
6-cyclohexanecarbonyl-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
1-(1H-imidazol-2-ylmethyl)-4-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,4-diazepane-6-carboxylic acid
N-({7-[2-(2,5-dimethoxyphenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
N-[2-(diethylamino)ethyl]-1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-methyl-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
(4aR,8aS)-1-[2-(2-fluorophenyl)ethyl]-6-(5-methylthiophene-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
(3S,4R)-4-(3-methoxyphenyl)-1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidine-3-carboxylic acid