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5-cyclopropanecarbonyl-1'-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(thiophen-2-yl)propan-1-one
(1R,5S,6S)-6-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
1-(3-ethyl-1,2-oxazole-5-carbonyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(1,4-dioxan-2-ylmethyl)-N,5-dimethyl-1H-pyrazole-4-carboxamide
N-cyclohexyl-3-({[(5-ethylfuran-2-yl)methyl]amino}methyl)-N-methylpyridin-2-amine
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-3-yloxy)ethyl]amine
4-(1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine-3-carbonyl)morpholine
N-{[7-fluoro-5-(quinolin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
N-(3-methylpyridin-2-yl)imidazo[1,2-a]pyrimidine-2-carboxamide
2-cyclopropyl-9-[(2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)ethyl]-1-methylpiperidine
5-[(4-methanesulfonylphenyl)methyl]-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
7-[(2S)-2-methoxy-2-phenylacetyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[2-({[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenoxy]-1-(4-methylpiperidin-1-yl)ethan-1-one
(2S)-1-(4-{[(2-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidine-2-carboxamide
1-(2-oxo-2-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethyl)piperidin-2-one
4,6-dimethyl-3-[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
5-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}-N-(furan-3-ylmethyl)thiophene-2-carboxamide
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-(propan-2-yl)-1H-pyrazole
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
2-(2,5-dioxoimidazolidin-1-yl)-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)acetamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
ethyl 2-{2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-1,3-oxazole-4-carboxylate
1-{2-[4-(hydroxymethyl)phenyl]acetyl}-3-(2-methoxyethyl)piperidine-3-carboxylic acid
(1R,5R)-6-[(2,3-dimethoxyphenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
methyl 5-{[4-(methylsulfamoyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
3-ethyl-1-({1-[(2-hydroxy-7-methylquinolin-3-yl)methyl]pyrrolidin-3-yl}methyl)urea
N-{4-[(2R)-2-methoxy-2-phenylacetamido]phenyl}-4-methylbenzamide
N-methyl-1-(2-phenylethyl)-N-{2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}piperidin-4-amine
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(1-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
N-(propan-2-yl)-1-[(1s,4s)-4-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,2-dihydroquinolin-2-one
3-chloro-4-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}phenol
2-(3-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}propyl)pyridine
N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
3-(2-methoxyethyl)-3-(1-methylpiperidin-4-yl)-1-(5-methylpyridin-3-yl)urea
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
2-(ethylamino)-N-[furan-2-yl(phenyl)methyl]pyrimidine-5-carboxamide
2-{4-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]morpholin-3-yl}acetamide
4-(5-butyl-4-phenyl-1H-imidazol-2-yl)pyrrolidin-2-one
1-(1,2,5-thiadiazole-3-carbonyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
4-cyclohexyl-N-(1,3,4-thiadiazol-2-yl)-1,4-diazepane-1-carboxamide
9-[(3-fluoro-2-methylphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
9-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-[(2-fluorophenyl)methyl]-1-(2-methoxyethyl)urea
5-methyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-[1-cyclohexyl-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-2-yl]ethan-1-ol
N-(2-oxopyrrolidin-3-yl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide