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1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
6-cyclopentyl-2-methoxy-3-[({thieno[2,3-d]pyrimidin-4-yl}amino)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-{4-[(2-methoxynaphthalen-1-yl)methyl]morpholin-3-yl}acetic acid
(2R,6R)-4-(1H-imidazol-4-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-tert-butyl-4-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
2-amino-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)pyridine-4-carboxamide
(2S,4R)-4-amino-N-methyl-1-(5-methylpyridine-3-carbonyl)pyrrolidine-2-carboxamide
1-{3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}pyrrolidin-3-amine
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N,1,3-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-N,N-dimethylpropane-1-sulfonamide
1-(1-{[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-4-phenylpiperidin-4-yl)ethan-1-one
2-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]-2-oxoethyl}-2-azaspiro[4.5]decan-3-one
1-{2-[(4aS,7aR)-4-methyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethyl}-2-methyl-1H-indole-3-carbonitrile
4-({2-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]phenyl}methyl)-1-methylpiperazin-2-one
2-(methylamino)-N-[2-(pyridin-2-yl)ethyl]pyridine-4-carboxamide
N-{2-[1-(3-hydroxypropyl)-4-phenyl-1H-imidazol-5-yl]quinolin-6-yl}acetamide
1-{2-methyl-2,8-diazaspiro[4.5]decane-3-carbonyl}-4-(pyridin-3-yl)piperidin-4-ol
5-[2-(2-methylpropoxy)phenyl]-1-propyl-1H-1,2,4-triazole
ethyl 1-(3-chloro-4-fluorobenzenesulfonyl)-4-(cyclopropylmethyl)piperidine-4-carboxylate
6-{3-[(2-fluorophenyl)methoxy]phenyl}-N,N-dimethylpyridine-3-carboxamide
2,5-dimethyl-3-{3-[(E)-2-phenylethenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrazine
1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
1-[3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)benzenesulfonyl]piperidine-3-carbonitrile
1-[3-(morpholine-4-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(2,3,6-trifluorophenyl)ethan-1-one
N-[(3R,4S)-4-cyclopropyl-1-(2-phenoxyacetyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
methyl 2-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl]piperidine-1-carboxylate
1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
6-[4-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carboxamide
dimethyl(2-{[5-(morpholine-4-carbonyl)furan-2-yl]oxy}hex-5-en-1-yl)amine
ethyl 4-[3-(benzylcarbamoyl)-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]piperidine-1-carboxylate
2,2-dimethyl-6-{3-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-3,4-dihydro-2H-pyran-4-one
2-[1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazol-4-yl)-N-methylformamido]-N-methylacetamide
1-cyclopentyl-5-(furan-2-yl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
2-cyclobutanecarbonyl-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-3-(3-fluorophenyl)propan-1-one
3-butyl-1-methyl-4-(6-methylpyridine-2-carbonyl)piperazin-2-one
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
N-(6-methylpyridin-3-yl)-3-[(2-oxopyrrolidin-3-yl)sulfamoyl]benzamide
2-(4-chlorophenyl)-4-(2-methoxy-3-methylbenzoyl)morpholine
3-(3-hydroxy-3-methylbutyl)-N-[(3S)-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl]benzamide
N2,N2-dimethyl-N4-[1-(pyridin-3-yl)ethyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
propan-2-yl 1-methyl-4-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
3-[2-(piperidin-2-yl)ethyl]-5-(pyrazin-2-yl)phenol
N-[2-(piperidin-1-ylmethyl)phenyl]-4-(pyridin-2-yl)piperazine-1-carboxamide
5-(2,5-dimethoxyphenoxy)-1-azabicyclo[3.2.1]octane
5-fluoro-N-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
N-(2-methoxyethyl)-6-(methoxymethyl)-N-[(2-methylphenyl)methyl]pyridine-2-carboxamide
4-methoxy-2-[2-(3-methoxyphenoxy)ethyl]pyrimidine
3-[2-(azocan-1-yl)-2-oxoethyl]-4-[(3-fluorophenyl)methyl]piperazin-2-one
N-{[4-(methylsulfanyl)phenyl]methyl}-N-propyl-3-(1H-1,2,4-triazol-1-yl)propanamide