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2-chloro-6-fluoro-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)benzamide
2-methyl-6-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]-3,4-dihydroquinazolin-4-one
N'-(4-methylphenyl)-N-{3-[(pyridin-3-yl)amino]propyl}propanediamide
N-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
4-(4H-1,2,4-triazol-4-yl)-1λ6-thiane-1,1-dione
1-(4-chlorophenyl)-N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
N-[(3S,4R)-1-(1H-indazole-3-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
2-amino-N,6-dimethyl-N-{[2-(trifluoromethyl)phenyl]methyl}pyrimidine-4-carboxamide
1-[2-({[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}amino)pyrimidin-4-yl]piperidin-3-ol
4-{2-[(6-ethyl-2-methylpyrimidin-4-yl)oxy]hex-5-en-1-yl}thiomorpholine
3-{[4-(3-fluorophenoxy)piperidin-1-yl]methyl}pyridine
8-[3-(3-chlorophenyl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
(2S)-3-phenyl-2-[4-(1-propyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propanamide
2-methyl-1-[2-(1-methylpiperidin-2-yl)ethyl]-1,4-dihydroquinolin-4-one
1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-pyrazol-1-yl)propan-1-one
N-methyl-N-(3-methylbutyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]urea
4-(2-fluoro-5-methylphenoxy)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylic acid
4-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidine-1-carbonyl)pyridine
2-methoxy-N-{[1-(quinolin-8-ylmethyl)pyrrolidin-3-yl]methyl}acetamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-N'-(3-ethylphenyl)butanediamide
5-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
7-(5-methyl-4-phenylthiophene-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methylpropanamide
(4aS,8aS)-2-(morpholine-4-sulfonyl)-decahydro-2,7-naphthyridin-4a-ol
4-cyano-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrrole-2-carboxamide
{3-[(3-methoxyphenyl)methyl]-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl}methanol
(4aR,7aS)-1-(furan-3-ylmethyl)-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-chlorophenyl)-1-(3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
1-(2-methoxyacetyl)-N-[2-(pyrrolidin-1-yl)ethyl]piperidine-3-carboxamide
6-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]pyrimidin-4-ol
N-[2-(3,4-dimethylphenoxy)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
3-methyl-1-[(3-methylphenyl)methyl]-4-(oxane-4-carbonyl)piperazin-2-one
(3aR,6aR)-2-benzyl-N-methyl-N-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-(4-methylpyrimidine-5-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5-{5-[(1-ethenyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2,1,3-benzothiadiazole
N-(2-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-2-yl}ethyl)acetamide
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[2-(pyridin-3-yl)piperidin-1-yl]propan-1-one
3-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene
4-(1-benzofuran-5-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
4-[4-(1H-imidazol-2-ylmethyl)piperazin-1-yl]-6-[(4-methylphenyl)sulfanyl]pyrimidin-2-amine
N6-benzyl-N5-[2-(1H-imidazol-1-yl)ethyl]-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-(1-methyl-1H-pyrrol-3-yl)-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)acetamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-7-fluoro-2-oxo-1,2-dihydroquinoline-4-carboxamide
4-ethyl-1-methyl-3-({1-[(3-methyl-1,2-benzoxazol-5-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[2-(morpholin-4-yl)ethyl]-3-[1-(1-phenylethyl)-1H-pyrazol-5-yl]urea
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,1-dimethyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
ethyl 2-[4-(4-fluorobenzenesulfonyl)-1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl]acetate