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1-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-4-(piperidin-1-yl)butan-1-one
4-[1-(3-fluorophenyl)-5-(morpholin-2-yl)-1H-1,2,4-triazol-3-yl]benzamide
[2-(4-ethylphenyl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
5-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole
1-[(3-methoxyphenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
1-(azocan-1-yl)-3-[5-({[2-(1H-imidazol-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-1,1-dioxo-1λ6-thiane-4-carboxamide
4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-2-one
4-[(prop-2-en-1-yl)sulfamoyl]-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]benzamide
2-(4-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperazin-1-yl)pyrimidine
5-(2-{[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]-N-methylbenzene-1-sulfonamide
ethyl 4-{3-[(4-methoxyphenyl)methyl]-1-methyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}piperidine-1-carboxylate
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
(2R,3S,6R)-5-(1H-indol-5-ylmethyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
4-{1-[(5-chloro-2,3-dimethoxyphenyl)methyl]azetidin-3-yl}morpholine
N4-[(1S)-1-carbamoyl-2-(4-hydroxyphenyl)ethyl]-N1,N1-dimethylpiperidine-1,4-dicarboxamide
(3S,4R)-1-(1H-indazole-3-carbonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)urea
1-(4-methyl-1H-imidazole-5-carbonyl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-methyl-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-phenylpiperazine
2-methyl-5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
3-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-(piperidin-4-yl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyrazine
6-(azepan-1-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
2-({1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidin-3-yl}formamido)-N,N-dimethylacetamide
3-(3-fluorophenyl)-N-[3-(1H-indazol-1-yl)propyl]-1H-pyrazole-4-carboxamide
5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-2-(2-methylphenyl)-1,3-thiazole
2-[3-(furan-2-yl)propanoyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
8-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(4-{[2-(furan-2-yl)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
(2S,4S,5R)-5-(2-fluorophenyl)-4-{[(3-hydroxyphenyl)methyl](methyl)carbamoyl}-1-methylpyrrolidine-2-carboxylic acid
(2R,6R)-11-methoxy-4-[(5-methylfuran-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[2-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazol-4-yl)ethyl]acetamide
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(dimethylamino)ethyl]-N-methylpropanamide
1-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
3-methyl-8-[3-(1H-pyrrol-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-[(4-chlorophenyl)methyl]-3-(1,3-dihydro-2-benzofuran-5-yl)-1-(3-hydroxypropyl)urea
4-benzyl-3-ethyl-1-(quinoxaline-5-carbonyl)-1,4-diazepan-5-one
(1S,5R)-6-(5-methyl-1,2-oxazole-3-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
dimethyl({4-methyl-5-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-[(2-chloropyridin-3-yl)methyl]-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
4-[(dipropylamino)methyl]-N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)benzamide
N-(oxan-2-ylmethyl)-3-[(1,2-oxazol-3-ylmethyl)sulfamoyl]benzamide
N-[(2-chlorophenyl)methyl]-5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carboxamide
N-methyl-N-[1-(pyrazin-2-yl)propan-2-yl]-4-sulfamoylbenzamide
4-(4-fluorophenyl)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1,2,3,6-tetrahydropyridine