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N-[2-(5-methylfuran-2-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(4aS,7aR)-1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-4-[3-(methoxymethyl)pyrrolidin-1-yl]-7-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
4-{5-[1-(dimethyl-1H-1,2,4-triazol-1-yl)propan-2-yl]-3-phenyl-1H-1,2,4-triazol-1-yl}-3-methylpyridine
1-{1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}azepane
4-{2-amino-3-cyano-5H,6H,7H-pyrrolo[2,3-h]quinolin-4-yl}-1-methyl-1H-pyrrole-2-carbonitrile
2-{4-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-1H-pyrazol-1-yl}-N-(1-methyl-1H-indazol-3-yl)acetamide
ethyl 1-(benzylsulfamoyl)piperidine-3-carboxylate
methyl({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})[1-(pyridin-2-yl)propyl]amine
1-(furan-3-carbonyl)-4-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-1,4-diazepane
5-{2-[(dimethylamino)methyl]phenyl}-N-methyl-4-(4-methylphenyl)pyrimidin-2-amine
5-[butyl(methyl)amino]-1-(cyclohexylmethyl)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{2-[(4-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperazin-1-yl)methyl]phenyl}methanol
2-{1-benzyl-4-[(3-ethoxy-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-({7-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1,3-diazinane-2,4-dione
1-(3-methoxypropanoyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
5-methoxy-2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,4-dihydropyridin-4-one
(2S,4R)-N-ethyl-4-[(1-methylpiperidin-4-yl)amino]-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
1-ethyl-4-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazine
4-(5-chloro-2-methylphenyl)-3-cyclobutyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-3-(pyridin-3-yl)propanamide
N-[1-(methylcarbamoyl)cyclohexyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-{3-[(4-chlorophenyl)sulfanyl]propyl}-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
1'-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(piperidine-1-carbonyl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
2-{[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}quinolin-4-ol
5-[1-(4-fluorophenyl)-2,2-dimethylcyclopropyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
5-oxo-1-phenyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,5-dihydro-1H-pyrazole-3-carboxamide
(1R,5S,6R)-3-[(1S,4S)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-N-[2-(1H-imidazol-4-yl)ethyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
(3R,4R)-3-cyclobutyl-1-{[3-(2-hydroxyethoxy)phenyl]methyl}-4-methylpyrrolidin-3-ol
1-[2-(2-fluoro-4-methylphenyl)pyrimidin-4-yl]piperidin-3-ol
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
5-{1-[(3S,4R)-3-benzyl-1-methylpiperidin-4-yl]-1H-1,2,3-triazol-4-yl}-2-methoxypyridine
N-(pyridin-3-ylmethyl)-3-{1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}propanamide
2-(cyclopropylmethyl)-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[5-(2-ethoxyethyl)-1,3,4-thiadiazol-2-yl]-3-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)urea
3-[({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)methyl]-1λ6-thiolane-1,1-dione
N-[2-(4-chlorophenyl)ethyl]-5-ethyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
1-{imidazo[1,2-b]pyridazin-6-yl}-4-(1,3-thiazol-4-ylmethyl)piperazine
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-{3-[4-(methylsulfanyl)phenyl]-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl}-2-azabicyclo[2.2.1]heptane
{6-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]pyridin-2-yl}methanol
N-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-4-yl)pyrimidin-2-amine
5-ethyl-6-methyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}thieno[2,3-d]pyrimidin-4-amine
1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)piperidine-3-carbonitrile
2-[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-methyl-N-phenylacetamide
methyl 2-[3-(2-{[(3,4-difluorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carbonyl]benzoate