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1-(isoquinolin-5-yl)-3-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}urea
3-hexyl-8-(4-methyl-1H-imidazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenol
4-benzyl-3-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[3-(propan-2-yloxy)propyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(3-methylphenyl)sulfanyl]piperidine
1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}-N-methylpiperidin-4-amine
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
2-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
2-[4-(4-fluorophenyl)-2-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy]-1-[2-(pyridin-3-yl)piperidin-1-yl]ethan-1-one
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-ethylacetamide
7-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-[4-(4-chlorobenzoyl)piperazin-1-yl]-2-[2-(3,4-dimethoxyphenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
1-[(2-fluorophenyl)methoxy]-8-(3,4,5-trimethoxybenzoyl)-1,8-diazaspiro[4.5]decan-2-one
N-methyl-1-[(E)-2-phenylethenesulfonyl]-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-(1H-imidazol-2-yl)piperidine
1-{4-[methyl(1,2-oxazol-3-ylmethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}cyclopropane-1-carbonitrile
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-1,3,7-trimethyl-1H-indole-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
ethyl 2-[({3-[2-hydroxy-3-(4-methylpiperazin-1-yl)propoxy]-4-methoxyphenyl}methyl)(methyl)amino]acetate
1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(pyrazin-2-yl)acetamide
8-cyclopropanecarbonyl-2-(1-ethyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-3-carbonyl}pyridine
3-{[1-(3,3-dimethylbutyl)piperidin-4-yl]methyl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(2-methylphenyl)acetamide
N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-2-(trifluoromethyl)pyrimidin-4-amine
9-(1,2-oxazole-3-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-6-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
1-ethyl-4-({4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)pyrrolidin-2-one
1-[2-(2-methyl-1H-imidazol-1-yl)propanoyl]-4-phenoxypiperidine-4-carboxylic acid
1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-3-[2-(2,4-difluorophenyl)ethyl]piperidine
1-{6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidin-4-yl}piperidin-4-ol
6-(hydroxymethyl)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)-1,4-oxazepane-4-carboxamide
8-(furan-3-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(4aR,7aS)-4-[(2,3-difluorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2-[(3-fluorophenyl)methyl]-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}morpholine
(3R,4R)-1-(1H-indole-6-carbonyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
(2R,3S)-2-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-3-hydroxybutanoic acid
2-(methylamino)-N-[2-(3-phenylpiperidin-1-yl)ethyl]pyrimidine-5-carboxamide
4-methyl-4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-chloro-5-acetamido-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]benzamide
N,1-dimethyl-N-[3-(oxolan-2-yl)propyl]-3-phenyl-1H-pyrazole-5-carboxamide
(2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-1-methyl-4-(morpholine-4-carbonyl)pyrrolidine-2-carboxylic acid
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
5-(3-chlorophenyl)-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-1,2,4-triazin-3-amine
7-[1-(3-hydroxypropyl)-4-phenyl-1H-imidazol-5-yl]-4-methyl-2H-chromen-2-one