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1-[(6-fluoroquinolin-2-yl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
3-[1-(1-phenylethyl)-1H-pyrazol-5-yl]-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}urea
1-ethyl-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(2-chlorophenyl)-4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
N-(2,3-dihydro-1H-inden-2-yl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
methyl 2-[4-(pyridin-4-yl)piperidine-1-carbonyl]piperidine-1-carboxylate
3-{5-[(3,4,5-trimethoxyphenyl)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
2-(5-chloro-2-methoxyphenyl)-2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]acetic acid
(benzylsulfamoyl)[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]amine
N-butyl-N-(furan-2-ylmethyl)-2,4-dimethylpyrimidine-5-carboxamide
1-[4-(3-fluorophenyl)phenyl]-3-[3-(4-methylpiperazin-1-yl)propyl]urea
2-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide
N-{2-[methyl(phenyl)amino]propyl}-1H-indazole-3-carboxamide
2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-methylazepane
5-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-cyclobutyl-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-benzyl-5-(4-benzylpiperidine-1-carbonyl)-N-ethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-(3-methylpyridin-2-yl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(pyrrolidin-3-yl)benzamide
2-oxo-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2,3-dihydro-1H-imidazole-4-carboxamide
methyl 3-(4-{[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
N-(2-{4-[(2-fluorophenyl)methyl]morpholin-2-yl}ethyl)methanesulfonamide
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]({[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl})methylamine
3-(2H-1,3-benzodioxol-5-yl)-1-[2-(4-methylpentyl)morpholin-4-yl]propan-1-one
6-acetyl-2-amino-4-[2-(5-methylfuran-2-yl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3E)-1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)pent-3-en-1-one
1-methanesulfonyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}piperidin-4-amine
3-benzyl-4-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazin-2-one
3-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1-(oxan-4-yl)piperidine
5-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]pyridine-2-carbonitrile
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(5-methyl-1H-1,2,4-triazol-3-yl)propanamide
2-methyl-4-{4-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]phenyl}butan-2-ol
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine
5-(2-phenylphenyl)pyridine-3-carboxamide
2-[3-methyl-4-(6-methyl-4-oxo-4H-chromen-3-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl]acetic acid
2-(dimethylamino)-2-(3-methylphenyl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
1-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
3-[({[2-(2-methylphenoxy)pyridin-3-yl]methyl}carbamoyl)methyl]-1,2,3-oxadiazol-3-ium-5-olate
4-(1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}piperidine-3-carbonyl)morpholine
2-(4-methylpentyl)-4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]morpholine
2-(cyclohex-1-en-1-yl)-1-[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
2-(2-chloro-4-fluorobenzenesulfonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
({2-[(dimethylamino)methyl]phenyl}methyl)(1H-imidazol-4-ylmethyl)methylamine
1-(4-cyclohexyl-1,4-diazepan-1-yl)-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
N-[(1-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-hydroxyazepan-4-yl)methyl]acetamide
4,6,7-trimethyl-2-{4-[2-(1,3-thiazol-2-yl)piperidin-1-yl]piperidin-1-yl}quinazoline
5-(oxolan-2-yl)-N-[2-(quinolin-8-yloxy)ethyl]thiophene-2-carboxamide
1-{2-[3-(1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
1-tert-butyl-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-5-oxopyrrolidine-3-carboxamide