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1-[1-(6-aminopyrimidin-4-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-(4-phenylbutyl)propanamide
2-({methyl[(1-phenylpyrrolidin-3-yl)methyl]amino}methyl)pyridine-3-carboxylic acid
4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-2,8-dimethylquinoline
11-(3-methoxybenzoyl)-4-[(2E)-2-methylbut-2-en-1-yl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
(3R,4R)-1-(6-methoxypyrimidin-4-yl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
4-({2-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(3-methoxypropyl)-2-methyl-N-{[2-(3-methylphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-1,3-thiazole-4-carboxamide
7-methyl-3-({methyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,7-dimethyl-1H-indole
N-benzyl-N-methyl-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-amine
7-methanesulfonyl-2-{4-[2-(2-methoxyphenyl)pyrrolidin-1-yl]piperidin-1-yl}-4-methylquinazoline
3-[1-(2-oxopropanoyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
[(3R,4R)-1-(5-methyl-1,2-oxazole-3-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-(3-hydroxypropyl)-9-(pyrimidin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-fluoro-5-methanesulfonamidophenyl)-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
2-ethyl-8-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
2-benzyl-4-(thiophene-3-carbonyl)morpholine
3-{1-[(2S)-1-acetylpyrrolidine-2-carbonyl]piperidin-4-yl}-N-benzyl-N-methylpropanamide
N-[(3R,5S)-1-cyclobutanecarbonyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
2-(naphthalen-1-ylmethyl)-4-(oxan-4-yl)morpholine
7-(1-benzothiophen-3-yl)-4-(1H-1,2,4-triazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-(cyclopropylmethyl)-1-methyl-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-({methyl[1-(3-methylpyridin-2-yl)propan-2-yl]amino}methyl)benzoic acid
N-[2-(4-{[3-(1,3-benzoxazol-2-yl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]cyclobutanecarboxamide
1-[7-(1,3-benzothiazol-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-phenyl-1,3-thiazol-4-yl)ethan-1-one
N-benzyl-N-methyl-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-amino-4-methyl-N-{2-[1-(2-methylpropyl)piperidin-3-yl]ethyl}pyrimidine-5-carboxamide
1-(1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}azetidin-3-yl)-2-methylpiperidine
3-methyl-N-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}benzamide
6-(propan-2-yl)-N4-[1-(pyrazin-2-yl)piperidin-3-yl]pyrimidine-2,4-diamine
(3aR,6aR)-N-[(2,3-difluorophenyl)methyl]-2-(2-methoxyacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-fluoro-3-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
1-methyl-4-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine-1-carbonyl}piperazine
5-(3-methoxyphenyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)furan-2-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-(1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}azetidin-3-ol
N-ethyl-N'-(2-fluoro-5-methylphenyl)-N-(oxolan-2-ylmethyl)butanediamide
3-(furan-2-yl)-3-phenyl-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-amine
2-amino-6-(2-methylpropyl)-N-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}pyrimidine-4-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(1-hydroxycyclopentyl)ethyl]-N-methylacetamide
9-(cyclopropylmethyl)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(cyclopropylmethyl)-N-propyl-1H-pyrazole-4-carboxamide
8-(5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-[3-(dimethylcarbamoyl)pyridin-2-yl]benzoic acid
N-[(1R,3R)-3-aminocyclopentyl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-[(5-methyl-1H-imidazol-4-yl)methyl]-4-(piperidin-3-yl)benzamide