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1'-[(2-fluoro-4-methoxyphenyl)methyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
5-butyl-1'-(1-methyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2-oxopiperidin-1-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
2-methyl-4-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidine-1-carbonyl}phenol
(4aS,8aS)-2-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-decahydro-2,7-naphthyridin-4a-ol
1-(cyclohexylmethyl)-N-[(2,3,4-trimethoxyphenyl)methyl]piperidin-3-amine
2-[4-(dimethyl-1,3-thiazole-5-carbonyl)piperazin-1-yl]-N-ethylacetamide
4-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-1-methyl-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decane
(2S,4R)-4-amino-N,N-diethyl-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}pyrrolidine-2-carboxamide
4-(piperidin-1-yl)-1-[(5-propylfuran-2-yl)methyl]piperidine-4-carboxamide
N-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(trifluoromethyl)benzamide
7-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(3S,4S)-1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
N-[(2R)-1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1-oxopropan-2-yl]acetamide
(3R,4R)-3-cyclopropyl-1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-methylpyrrolidin-3-ol
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-methyl-2,3-dihydro-1H-indene-2-carboxamide
(1S,5R)-6-[(dimethylcarbamoyl)methyl]-N-(4-methoxyphenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N3-[3-(dimethyl-1,3-thiazol-2-yl)propyl]piperidine-1,3-dicarboxamide
2,4-dimethyl-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)pyrimidine-5-carboxamide
6-methyl-N-[(4-sulfamoylphenyl)methyl]imidazo[2,1-b][1,3]thiazole-5-carboxamide
1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-5-(1,3-thiazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(oxolan-2-ylmethyl)-2-{2-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
N,N-dimethyl-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]pyrrolidin-3-amine
5-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-2,4-dimethylpyrimidine
5-(4-fluorophenyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidine-1-carbonyl]naphthalen-2-ol
1-[benzyl(methyl)amino]-3-[4-(thiomorpholin-4-ylmethyl)phenoxy]propan-2-ol
1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-[4-(oxolan-2-yl)butyl]urea
N-ethyl-2-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}acetamide
(3-methyl-1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methanol
2-methyl-6-{2-[(2E)-4-methylpent-2-en-1-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
2-{4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}ethan-1-ol
ethyl 4-[1-(2-cyclopentyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-3-carbonyl]piperazine-1-carboxylate
benzyl N-(1-{[2-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl)carbamate
2-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
8-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]thiophene-3-sulfonamide
3-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-N-(propan-2-yl)propanamide
6-hydroxy-2,5,7,8-tetramethyl-N-(pyrimidin-4-ylmethyl)-3,4-dihydro-2H-1-benzopyran-2-carboxamide
1-[6-(2,3-dimethoxyphenyl)pyridazin-3-yl]azepane
1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-cyclopropyl-3-ethoxy-4-(prop-2-en-1-yloxy)-N-(pyridin-3-ylmethyl)benzamide
3-(3-chlorophenyl)-3-phenyl-N-[2-(pyridin-3-yl)ethyl]propanamide
2-(2-chlorophenyl)-5-methyl-4-[(4-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
(2S,4S)-4-amino-1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3R,5S)-N-[(4-chlorophenyl)methyl]-1-(pyridin-3-ylmethyl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
2-[6-hydroxy-4-(quinoxalin-2-yl)-1,4-diazepan-1-yl]pyridine-3-carbonitrile
2-(3-chlorophenoxy)-1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
6-[3-(1-methoxyethyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile