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methyl (2S,4R)-1-(naphthalen-1-ylmethyl)-4-[2-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
1-[(1R,5S,6R)-6-{[4-(2-propoxyethyl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexan-3-yl]ethan-1-one
3-cyclopropyl-5-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-3-(methoxymethyl)piperidine
1-(2-{1-[(4-acetamidophenyl)methyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[(3S,4R)-1-(3-methoxypyrazin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-cyclopropanecarbonyl-N-[4-(2-fluorophenoxy)phenyl]piperidine-4-carboxamide
2-{[1-(3-methylpyridin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}morpholine
3-{4-[2-(benzyloxy)ethyl]piperazin-1-yl}pyrazine-2-carbonitrile
4-[2-(3-cyclopropanecarbonyl-1H-indol-1-yl)acetyl]-1λ6-thiomorpholine-1,1-dione
1-methyl-4-[3-(thiomorpholine-4-carbonyl)benzenesulfonyl]piperazin-2-one
4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-3,3-dimethylpiperazin-2-one
2-(2-aminoethyl)-N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]quinazolin-4-amine
(3S,5R,9R)-N-benzyl-5-hydroxy-2,8-dioxo-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-11-carboxamide
1-[1-(furan-2-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-(3-methyl-1,2-oxazol-5-yl)-1-[4-(pyrazin-2-yl)piperazin-1-yl]ethan-1-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-oxo-1,4-dihydroquinoline-2-carboxamide
ethyl 1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-4-(2-phenylethyl)piperidine-4-carboxylate
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(3R,4R)-4-hydroxy-1-methyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}piperidine-3-carboxamide
7-fluoro-3-methyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1-benzofuran-2-carboxamide
N-cyclopropyl-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperazine-2-carboxamide
5-{2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[3-(furan-2-yl)benzoyl]-4-(2-methylpropyl)-1,4-diazepan-5-one
N-ethyl-N-(oxan-4-ylmethyl)-3-propanamidobenzamide
N3-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-N1,N1-dimethylpiperidine-1,3-dicarboxamide
4-({3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
5-phenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,3,4-thiadiazol-2-amine
(3S,4S)-4-cyclopropyl-1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}pyrrolidine-3-carboxylic acid
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
N-[1-(furan-2-carbonyl)piperidin-4-yl]-5-phenyl-1,2-oxazole-3-carboxamide
3-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-6-methoxy-1,4-dihydroquinolin-4-one
2-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline
N-({5-[(1-propyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
4-[5-(2-ethoxyphenyl)furan-2-carbonyl]morpholine
3-(1-methylpiperidin-3-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
2-amino-4-(piperidin-4-yl)-6-(1-propyl-1H-1,2,3-benzotriazol-5-yl)pyridine-3-carbonitrile
7-[2-(piperidin-1-yl)acetyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6-methoxy-N4-methyl-N4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidine-2,4-diamine
6-chloro-N-[(3-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)imidazo[1,2-a]pyridine-2-carboxamide
5-(3-ethoxyphenyl)pyridine-2-carbonitrile
N-[(1S,2R)-2-aminocyclobutyl]-2-(3-phenyl-1,2,4-oxadiazol-5-yl)benzamide
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N4-(propan-2-yl)pyrimidine-2,4-diamine
3-methoxy-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}propan-1-one
1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(1,3-dihydro-2-benzofuran-5-yl)-3-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
3-{2-[(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)amino]ethyl}-1,3-oxazinan-2-one
(2S,4R)-4-(4-{2-[(2-methoxyphenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
7-[2-(5-methylthiophen-2-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]propanamide