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(9aR)-2-methyl-8-(4-methylbenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(3-methoxypropyl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine-3-carboxylic acid
(3E)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}hex-3-enamide
3-({1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
1-(1H-indazol-7-yl)-3-methyl-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
(1S,5R)-6-[4-(propan-2-yl)benzoyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-5-(morpholin-4-ylmethyl)-N-[1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
ethyl 1-(5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)piperidine-3-carboxylate
9-(3,5-dimethylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)urea
3-ethyl-1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidine-3-carboxamide
N-[4-(1H-indol-2-yl)phenyl]-1-(2-methylbutanoyl)piperidine-4-carboxamide
7-chloro-3,5-dimethyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1-benzofuran-2-carboxamide
2-[(1H-imidazol-2-ylmethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]ethan-1-ol
5-methanesulfonyl-N-[(2-methylphenyl)methyl]-4-(piperidin-3-yl)pyrimidin-2-amine
methyl[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
1-[2-(3-fluorophenyl)piperidin-1-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
4-(cyclohexylmethyl)-3-(pyridin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
(1S,5R)-3-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1,3-thiazole-4-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)(2,1,3-benzoxadiazol-4-ylmethyl)(pyridin-3-ylmethyl)amine
1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1,4-diazepan-6-ol
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-[4-(2-ethoxyphenyl)piperazin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
(1R,4S)-2-(2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carbonyl)-2-azabicyclo[2.2.1]heptane
5-(dimethyl-1,3-thiazol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
7-(2H-1,3-benzodioxole-5-carbonyl)-N-(prop-2-en-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(3-chloropyridin-2-yl)-4-(2-phenoxyethyl)piperidine-4-carboxylic acid
6,8-dimethyl-2-{[4-(pyridin-4-ylmethyl)piperazin-1-yl]methyl}quinolin-4-ol
3-hydroxy-3-{[(1H-indol-6-ylmethyl)amino]methyl}-1-(3-phenylpropyl)piperidin-2-one
2-[2-(methylsulfanyl)pyrimidin-4-yl]-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
3-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
N,N-dimethyl-4-[2-(2-oxo-1,2-dihydroquinolin-1-yl)acetyl]piperazine-1-sulfonamide
3-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)propanamide
(3S,4R)-1-(1-methyl-1H-pyrrole-2-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidine-2-carboxamide
11-[(cyclopropylmethyl)amino]-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl 2-[butyl(methyl)sulfamoyl]-6-[(4-methoxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(5-chloro-2-methylphenyl)-4-(2-ethoxyethyl)piperazine
2-fluoro-6-({4-[4-(hydroxymethyl)pyridin-2-yl]piperazin-1-yl}methyl)phenol
3-{1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}benzonitrile
4-(5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)morpholine
1-{2-oxo-2-[2-(2-phenylethyl)morpholin-4-yl]ethyl}piperidin-2-one
3-{[methyl({[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amino]methyl}phenol
(4aR,7aS)-1-[2-(piperidin-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-propyl-3-({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}sulfamoyl)benzamide
N-[(3R,4S)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-4-propylpyrrolidin-3-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
N-(1-hydroxybutan-2-yl)-3-(pyrimidin-2-yloxy)-N-(thiophen-2-ylmethyl)benzamide
(1S,5R)-3-(oxan-4-yl)-6-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane