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6-(2-chlorophenyl)-7-methyl-2-(2-methylpyrrolidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
5-tert-butyl-3-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
N-{[5-(methylcarbamoyl)furan-2-yl]methyl}-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methylacetamide
N-{[7-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1H-indole-2-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}propanamide
1-(azocan-1-yl)-3-{4-[(cyclohexylamino)methyl]-2-methoxyphenoxy}propan-2-ol
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}amine
1-[2-methoxy-6-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}-3-methylpyrazine
4-(1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)morpholine
methyl (2R,4S)-4-hydroxy-1-[(3-hydroxy-6-methylpyridin-2-yl)methyl]piperidine-2-carboxylate
4-{4-[(4-ethoxyphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
5-({7-chloro-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[(2R,4R,6S)-2-tert-butyl-6-(2-cyclohexylpyrimidin-5-yl)oxan-4-yl]acetamide
N-(1-cyclopentanecarbonylazepan-3-yl)-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
5-benzyl-N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[2-(3-methoxyphenyl)phenyl]-1-(pyrimidin-2-yl)piperidine-4-carboxamide
methyl 9-(cyclopentyloxy)-7-oxo-3-(oxolane-3-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(2,3-dihydro-1-benzofuran-7-yl)-2-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]acetic acid
7-[2-(2-methylphenyl)acetyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
6-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]pyridin-2-amine
2-({[(3R,4R)-4-(hydroxymethyl)-1-(2-methylpyrimidin-4-yl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-(dimethylamino)-N-methyl-2-(4-methylphenyl)-N-(quinoxalin-2-ylmethyl)acetamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(2-oxopyrrolidin-1-yl)acetamide
N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-2-cyclopropylacetamide
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
N-phenyl-2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
N-[2-(morpholin-4-yl)ethyl]-2-[2-(propylsulfanyl)acetamido]benzamide
7-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-2,4-dimethylquinoline
1-[1-(2-phenylethyl)piperidin-4-yl]-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
1-[(1-benzyl-3-methyl-1H-1,2,4-triazol-5-yl)methyl]-4-ethylpiperazine
3-[5-(5-acetylthiophene-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-(furan-2-ylmethyl)-6,7-dimethoxy-3,4-dihydroquinazolin-4-one
N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-[3-(pyridin-3-yl)propanamido]cyclopentane-1-carboxylic acid
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N-(1,4-dioxan-2-ylmethyl)-N-methylpiperidin-4-amine
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
N-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2,5,6-trimethyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]pyrimidin-4-amine
3-(1-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}azetidin-3-yl)pyridine
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidine
2-{[4-(2-methoxyphenyl)-5-(3-methylthiophen-2-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
4-(2-oxopiperidin-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]butanamide
N-[2-(benzyloxy)ethyl]-1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-5-methanesulfonyl-2-methylpyrimidine
3-(1-benzylpiperidin-3-yl)-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-methyl-N-[3-(oxolan-2-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine