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N-[2-(azepan-1-yl)-2-phenylethyl]-2-(ethylamino)pyrimidine-5-carboxamide
8-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
N-[(2S)-1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(1H-imidazol-4-yl)-1-oxopropan-2-yl]acetamide
methyl 3-{[1-(cyclopropylmethyl)-5-(3-phenylprop-2-ynoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
(3S,4R)-4-(2-methoxyphenyl)-1-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]pyrrolidine-3-carboxylic acid
1-ethyl-5-methyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
4-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]-1-(2-methoxyphenyl)piperazin-2-one
4-chloro-1-methyl-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]-1H-pyrazole-5-carboxamide
3-ethyl-4-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}morpholine
1-(5-acetyl-2-methoxyphenyl)-3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]urea
1-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-(1H-imidazol-1-yl)-1-[(2-methoxy-4-methylphenyl)methyl]piperidine-4-carboxylic acid
5-{2-[(4aS,8aR)-1-butyl-2-oxo-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{[(2-methoxyphenyl)methyl]amino}-N,5-dimethyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(3,6-dimethylpyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-cycloheptyl-N-(1H-imidazol-2-ylmethyl)-N-methyl-6-oxopiperidine-3-carboxamide
1-(2-chlorophenyl)-4-(oxan-2-ylmethyl)piperazine
6-ethoxy-3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
3-chloro-2-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}pyridine
3-{[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]sulfamoyl}-N-methyl-N-(2-methylpropyl)benzamide
N-tert-butyl-1-cyclohexyl-5-(4-cyclopentylpiperazine-1-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]-2H-1,3-benzodioxole-5-carboxamide
N-[(2R)-1-hydroxy-3-methylbutan-2-yl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
N-cyclopropyl-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)furan-3-carboxamide
N-[2,2-dimethyl-3-(morpholin-4-yl)propyl]-N-[(2-methoxyphenyl)methyl]cyclopropanamine
3-methyl-7-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(3aR,7aS)-2-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(1S,2S)-2-[4-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]cyclohexan-1-ol
3-amino-1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)pyrrolidine-3-carboxylic acid
N3-cyclooctyl-4-oxo-N5-(oxolan-2-ylmethyl)-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
5-(3-fluorophenyl)-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-1,2,4-triazine
ethyl 2-[2-(5-{[2-(1H-imidazol-1-yl)ethyl]carbamoyl}thiophen-2-yl)pyrrolidin-1-yl]acetate
(3aS,6aS)-2-(4-chloro-3-fluorobenzoyl)-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(4aR,8aS)-1-(thiophen-2-ylmethyl)-decahydro-1,6-naphthyridin-6-yl]-2-phenoxyethan-1-one
3-[(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)amino]-2,3-dihydro-1λ6-thiophene-1,1-dione
7-(2-hydroxy-5-methoxybenzoyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-2-yl)pyridine
N-[(5-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
6-{3-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
3-{[1-(3-cyano-2-methoxypyridin-4-yl)pyrrolidin-3-yl]methyl}benzamide
N-butyl-4-cyano-N-[(3-methoxyphenyl)methyl]benzamide
(1R,3S,5S)-8-{2-[(prop-2-en-1-yl)amino]benzoyl}-8-azabicyclo[3.2.1]octan-3-ol
1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
N-(2-hydroxyethyl)-3-{5-[3-(1-methyl-1H-pyrrol-2-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-cyclopropanecarbonyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxamide
(3R,5S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
(2S,4S,5R)-4-(butylcarbamoyl)-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
N-methyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide