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N-{1-[({[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}-3-phenoxypropanamide
1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4-(morpholin-4-yl)pentan-1-one
(3R,4R)-1-[(1-benzyl-1H-indol-6-yl)methyl]-4-(hydroxymethyl)piperidin-3-ol
2-{3-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
(3aR,6aR)-2-[5-(methoxymethyl)thiophene-2-carbonyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}azetidin-3-ol
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-(2-methoxyphenoxy)ethan-1-one
3-{imidazo[1,2-a]pyridin-2-yl}-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)propanamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-hydroxy-N-methyl-2-(thiophen-2-yl)pyrimidine-5-carboxamide
3-(3-methoxyphenyl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-(3-methylpyridin-4-yl)-4-(1,3-thiazol-2-ylmethyl)piperazine
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[2-(pyridin-3-yloxy)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
4-(4-methylpiperazin-1-yl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pentan-1-one
5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
(2S)-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}piperidine-2-carboxamide
1-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4,4-difluoropiperidine
3-[(4aR,7aS)-4-(5-methylthiophene-3-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
8-(2H-1,3-benzodioxole-5-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
N,4-dimethyl-2-(propan-2-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1,3-thiazole-5-carboxamide
4-{1-[5-(propan-2-yl)thiophene-3-carbonyl]piperazine-2-carbonyl}morpholine
2-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-methyl-1H-1,3-benzodiazole
(1S,5R)-3-(3-fluorobenzoyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-({4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
1,5-dibenzyl-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3aS,6aR)-5-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-[(1S,2S)-2-hydroxycyclohexyl]-N-(2-methyl-1-benzofuran-5-yl)piperazine-1-carboxamide
N-(4-fluorophenyl)-1-(6-methylquinoline-4-carbonyl)piperidin-3-amine
2-methanesulfonamido-N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]acetamide
2-(3-chloro-2,4-difluorophenyl)-1-(prop-2-en-1-yl)-1H-imidazole
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-N,N-bis(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aS,8aR)-1-(3-hydroxypropyl)-6-(thiophene-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclopropanesulfonamide
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(oxolan-2-ylmethyl){[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
2-(2-methylpropyl)-8-(3-phenyl-1,2-oxazole-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methoxyphenyl)ethan-1-one
methyl[(3-methyl-1H-indol-2-yl)methyl]{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
2-(4-chlorophenyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-[2-fluoro-3-(trifluoromethyl)phenyl]-5-(methanesulfonylmethyl)pyridine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2,6-difluoro-N-methylbenzene-1-sulfonamide
N-(3-methoxypropyl)-6-[2-(pyridin-2-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-ethyl-2-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
3-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-1-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
2-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-cyclopropyl-N-(1H-indol-5-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[4-(pyrrolidin-1-yl)butyl]acetamide
1-[(2-chlorophenyl)methyl]-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-{1-[4-(3-fluorophenyl)benzoyl]piperidin-4-yl}morpholine