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2-(phenylsulfanyl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
ethyl 3-{[1-(2-methoxyethyl)-6-oxopiperidin-3-yl]formamido}propanoate
(3aS,6aS)-2-[2-(2-ethylphenoxy)ethyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(2,4-dimethoxyphenyl)ethyl]-2-[methyl(piperidin-4-yl)amino]acetamide
3-(benzenesulfonyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]propanamide
3-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-[4-(ethylsulfanyl)phenyl]urea
2-(4-{5-[(phenylsulfanyl)methyl]furan-2-carbonyl}morpholin-3-yl)acetic acid
1-methyl-3-(1-methyl-1H-pyrazol-4-yl)-1-[3-(oxolan-2-yl)propyl]urea
1-(4-methoxyphenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]cyclopropane-1-carboxamide
4-[4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-yl]morpholine
1-(4-methylpiperazin-1-yl)-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)ethan-1-one
2-(azepan-1-yl)-N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-oxoacetamide
1-[5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidine-3-carboxamide
9-[(3,5-dimethoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-({[(2-fluorophenyl)methyl](2-methoxyethyl)amino}methyl)-2,6-dimethoxyphenol
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-3-azaspiro[5.5]undecan-9-amine
3-{[cyclopropyl({[2-(dimethylamino)pyrimidin-5-yl]methyl})amino]methyl}phenol
7-[3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-2-amino-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
3-(2-fluorophenyl)-1-[3-(methylsulfanyl)propyl]pyrrolidine
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]pyrrolidine-2-carboxamide
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
3-[1-(1H-indole-6-carbonyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(quinoxalin-2-yl)piperidin-3-amine
8-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-{1-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
2-(3-methoxyphenyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
8-methoxy-4-methyl-2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]quinoline
[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl][1-(4-methylpiperazin-1-yl)propan-2-yl]amine
N-(2-fluorophenyl)-2-{4-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetyl]morpholin-3-yl}acetamide
N,2-dimethyl-N-[3-(oxolan-2-yl)propyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
5-(hydroxymethyl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]furan-2-carboxamide
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pent-4-enamide
3-{[4-(2-aminopyrimidin-4-yl)piperidin-1-yl]methyl}-2,4-dichlorophenol
4-{4-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridine-2-carbonyl}morpholine
methyl (2R,4S)-4-hydroxy-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine-2-carboxylate
3-(4-{[3-hydroxy-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]methyl}piperazin-1-yl)pyrazine-2-carbonitrile
3-chloro-N-(2-methoxyethyl)-4-({1-[4-methyl-4-(methylsulfanyl)pentan-2-yl]piperidin-4-yl}oxy)benzamide
5-{methyl[(3-methylthiophen-2-yl)methyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-[(3-methoxyphenyl)methyl]-4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
6-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purin-2-amine
cyclopentyl 4-({[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]carbamoyl}amino)benzoate
{3-[(2-methylphenyl)methyl]-1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl}methanol
4-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-3-(2-hydroxyethyl)piperazin-2-one
4-[2-(2-chlorophenyl)ethyl]-11-[4-(2-methoxyethyl)piperazin-1-yl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-[7,8-dimethyl-2-(pyrimidin-5-yl)quinoline-4-carbonyl]-1,3-dimethylpiperazin-2-one
methyl (2S,4R)-4-(2,3-dimethyl-1H-indole-7-amido)-1-(3-phenylpropyl)pyrrolidine-2-carboxylate
1-{5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}azepane
3-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methoxy}pyridin-2-amine