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3-{[2-(3-fluorophenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-[2-(pyrrolidin-1-yl)ethyl]piperidine-3-carboxamide
3-methoxy-2-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenol
3-(dimethylamino)-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)benzamide
(3S,9aR)-8-[(2-fluoro-5-methylphenyl)methyl]-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N3-benzyl-1-cyclohexyl-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(5-methylpyridine-3-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-(6-methyl-5-{[(2-methylfuran-3-yl)formamido]methyl}-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carbonyl)-2,1,3-benzoxadiazol-1-ium-1-olate
3-ethyl-8-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
4-({2-[1-(3-chlorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-amine
2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]quinoline
ethyl 4-({2-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)piperazine-1-carboxylate
8-(cyclobutylmethyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
1,5-dimethyl-3-{[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]methyl}-1H-indazole
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
6-[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-9H-purine
1-ethyl-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-3-ylmethyl)acetamide
2-(dimethylamino)-7-[(1-ethyl-1H-imidazol-2-yl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-(4-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carbonyl}piperazin-1-yl)phenol
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]morpholine-2-carboxamide
N-benzyl-4-(1-hydroxy-2-phenylethyl)piperidine-1-sulfonamide
N-methyl-4-phenoxy-N-(1H-pyrazol-3-ylmethyl)butanamide
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-methoxypropan-1-one
N-[1-(1-acetylpiperidin-4-yl)-1H-pyrazol-5-yl]-1-phenylmethanesulfonamide
4-({4-methyl-5-[(oxan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)piperidine
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4-(1H-imidazol-1-yl)butan-1-one
4-{6-[3-(methylsulfanyl)phenyl]pyridine-3-carbonyl}morpholine
2-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-2,7-diazaspiro[4.5]decane
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-1,3-thiazole-4-carboxamide
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2-(trifluoromethyl)benzamide
ethyl 2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]pyridine-3-carboxylate
2-(2-methoxyethyl)-8-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-methyl-1,3-thiazole-4-carboxamide
(2S,4S)-4-acetamido-N-ethyl-1-{[3-(morpholin-4-yl)phenyl]methyl}pyrrolidine-2-carboxamide
3-cyclohexyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H-pyrazole-4-carboxamide
4-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-{3-[4-(cyclopropylmethyl)piperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol
(2S,4S)-1-benzyl-N-[2-(2-fluorophenyl)ethyl]-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-(pyridin-2-ylmethyl)acetamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(2-ethylpiperidin-1-yl)ethan-1-one
N-benzyl-5-(4-chloro-2-methoxyphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
1-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]cyclopropan-1-amine
1-(1-hydroxypropan-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-3-{[2-(2-hydroxyethyl)piperidin-1-yl]methyl}benzamide
(4aS,7aR)-1-[2-(benzyloxy)acetyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione