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3-methyl-4-({[2-(4-phenylpiperidin-1-yl)ethyl]carbamoyl}amino)benzamide
N-[3-(hydroxymethyl)-2-methylphenyl]-2-[4-(2-methyl-1,3-thiazole-4-carbonyl)morpholin-3-yl]acetamide
3-(diphenylmethyl)-5-methyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-5-methoxy-1H-indole
(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
1-(3-{[methyl(thian-4-yl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
4-[(1-cyclopentanecarbonylpiperidin-4-yl)oxy]-N-(2-phenylethyl)benzamide
3-methyl-5-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2-oxazole
1-methyl-6-oxo-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,6-dihydropyridazine-3-carboxamide
2-({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)-N-[1-(4-methylphenyl)ethyl]acetamide
8-(quinoline-3-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-({3-[(1H-indazol-5-yl)carbamoyl]phenyl}methyl)-N-methylpyrrolidine-3-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(naphthalen-2-yloxy)propanamide
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(1H-indol-3-yl)ethan-1-one
N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-3-yloxy)acetamide
(1S,5R)-6-(2-methoxyethyl)-3-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4R)-N-(1,3-dihydro-2-benzofuran-5-yl)-1-[(5-methylthiophen-2-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
4-(2-chloro-4-fluorobenzoyl)-1-(2-methylphenyl)piperazin-2-one
6-ethyl-2-{3-[(2-phenylmorpholin-4-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
7-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(azepane-4-carbonyl)-4-(4-fluoro-2-methylphenoxy)piperidine-4-carboxylic acid
4-[2-(3,4,5-trimethoxyphenyl)acetyl]morpholine-2-carboxylic acid
4-{3-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]propoxy}benzamide
N-[2-(1-methylpiperidin-3-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-imidazole
N-(2,5-dimethoxyphenyl)-3-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}propanamide
1-[4-(2-phenylethyl)piperazin-1-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
N-[3-(1H-imidazol-1-yl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
1-[(2,4-dimethoxyphenyl)methyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
9-[2-(propan-2-ylsulfanyl)acetyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-methoxyphenyl)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]cyclopentane-1-carboxamide
2-(4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-1,3-benzothiazole
3-(3-chlorophenyl)-3-{[1-(propan-2-yl)piperidin-4-yl]formamido}propanoic acid
1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-N-(furan-2-ylmethyl)piperidine-4-carboxamide
5-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-(2-methoxyethyl)-1,2,4-oxadiazole
1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-N-(3-methylbutyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2S,4R)-4-amino-N-methyl-1-[1-(2-phenylacetyl)piperidine-4-carbonyl]pyrrolidine-2-carboxamide
(2-{[4-(6-methylpyridazin-3-yl)piperazin-1-yl]methyl}phenyl)methanol
N-(furan-3-ylmethyl)-N-methyl-3-propyl-1H-pyrazole-4-carboxamide
(2R,3R)-1'-[(3-methyl-1H-pyrazol-5-yl)methyl]-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
{[4-(furan-3-ylmethyl)-1,4-oxazepan-6-yl]methyl}dimethylamine
(1R,2S,9R)-11-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
1-cyclopropanecarbonyl-N-{1-[4-(dimethylamino)phenyl]propan-2-yl}piperidine-4-carboxamide
(3S)-1,3-dimethyl-4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-ethyl-N-methyl-5-oxopyrrolidine-3-carboxamide
{4-methyl-5-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methanol
N-(adamantan-1-ylmethyl)-N-methyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine