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2,4-dimethyl-5-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,3-thiazole
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-chloro-3-fluoropyridine
(butan-2-yl)({[2-(4-methanesulfonylphenyl)phenyl]methyl})amine
ethyl 1-(2-hydroxyethyl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
1-(3-chlorophenyl)-4-(4,6-dimethylpyridine-3-carbonyl)piperazin-2-one
1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
2-(2H-1,3-benzodioxol-5-yloxy)-1-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propan-1-one
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-({[(5-chloro-3-methoxy-2-propoxyphenyl)methyl](methyl)amino}methyl)-1-methylpyrrolidin-2-one
2-(2-methoxy-4-{3-methyl-6-oxo-1-propyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}phenoxy)acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(3,3,3-trifluoropropyl)piperidine
2-({2-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]phenyl}amino)acetic acid
(2S,4R)-1-[2-(3-acetyl-7-ethyl-1H-indol-1-yl)acetyl]-4-amino-N-methylpyrrolidine-2-carboxamide
N-[cyclopropyl(4-methoxyphenyl)methyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({imidazo[1,2-a]pyrimidin-6-ylmethyl})methylamine
1-[1'-(2,5-dimethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
6-{1-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-3-yl}pyrimidin-4-ol
3-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
2-methyl-4-(piperidin-3-yl)-6-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidine
5-(2H-1,3-benzodioxol-5-yl)-3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
2-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(2S,4S)-4-amino-1-(cyclohex-1-ene-1-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
3-(2-{4-[hydroxy(phenyl)methyl]piperidin-1-yl}-2-oxoethyl)-3-(3-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
N,N-dimethyl-2-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)acetamide
(3S,4R)-4-(3-fluorophenyl)-1-(quinoxaline-6-carbonyl)pyrrolidine-3-carboxylic acid
1-benzyl-N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]pyrrolidin-3-amine
3-ethyl-1-(2-phenylethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[3-(1-methoxyethyl)phenyl]pyrimidin-4-yl}piperidin-4-ol
[(4-ethyl-5-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
(4aS,8aR)-6-(3-methoxypyrazin-2-yl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
N-(1,3-dihydroxypropan-2-yl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-ethoxy-3-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridine
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
3-({[(2-chloro-6-fluorophenyl)methyl]amino}methyl)-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
N-[2-phenyl-2-(piperidin-1-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyrrolidin-2-one
1-[2-methyl-3-(1H-pyrrol-1-yl)phenyl]-3-{[1-(morpholin-4-yl)cyclopentyl]methyl}urea
1-{2-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-oxoethyl}-2-methyl-1,4-dihydroquinolin-4-one
5-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-propyl-1H-pyrazole
3-{1-[3-(5-methylfuran-2-yl)butyl]azetidin-3-yl}pyridine
1-(1H-1,2,3-benzotriazole-5-carbonyl)azepan-4-amine
N-(furan-3-ylmethyl)-N-methyl-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-{3-[3-(5-acetyl-2-fluorophenyl)phenyl]-1H-pyrazol-1-yl}acetamide
5-fluoro-2-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
3-methoxy-1-{2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(4-fluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione