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N-cyclopentyl-1,3-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(5-methylpyrazin-2-yl)methyl]-9-(oxane-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-benzyl-N,5-dimethyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-(2-methoxyethyl)-2-(pyridine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
4-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]-N,N-dimethylbenzene-1-sulfonamide
7-(morpholine-4-sulfonyl)-2-[(2S)-oxolane-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
methyl 1-(cyclopropylmethyl)-3-{[5-(dimethylcarbamoyl)furan-2-yl]methyl}-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
8-methyl-3-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}-2-(thiophen-2-yl)quinoline
4-[(4-fluorophenyl)methyl]-1-(3-methylfuran-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-methyl-N-[(2-methylphenyl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
(3R)-1-[6-amino-2-(diethylamino)pyrimidin-4-yl]pyrrolidin-3-ol
2-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-6-methylpyrimidin-2-amine
N-benzyl-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N-methylpiperidin-4-amine
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
8-methoxy-4-methyl-N-[(2S)-oxolan-2-ylmethyl]quinolin-2-amine
N-tert-butyl-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)butanamide
5-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
N'-(4-methylphenyl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}propanediamide
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-[2-(diethylamino)ethyl]-5-(methoxymethyl)-N-methyl-1H-pyrazole-4-carboxamide
3-(cyclobutylsulfamoyl)-N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]benzamide
(3R,4S)-4-[methyl({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino]oxolan-3-ol
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-[2-(3-fluorophenyl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(butan-2-yl)[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl](pyridin-4-ylmethyl)amine
1-ethyl-3-{1-[2-(3-fluorophenyl)ethyl]-1H-imidazol-2-yl}piperidine
4-({5-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
N-{1-[1-(2-amino-2-methylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
N-(2-methylpropyl)-3-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-(thiophen-3-ylmethyl)propanamide
5-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(5-methyl-1,2-oxazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-2-methanesulfonylacetamide
N-[(1-benzyl-4-hydroxyazepan-4-yl)methyl]morpholine-4-sulfonamide
5-(4-cyclohexylphenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2,4-triazin-3-amine
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-(5-fluoropentyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
2-[(3-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)methyl]-1H-1,3-benzodiazole
(1-{5-[1-(oxan-4-ylmethyl)pyrrolidin-2-yl]thiophene-2-carbonyl}piperidin-4-yl)methanol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-propanamidopropanamide
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-({[(3R,4R)-1-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
4-(4-fluorophenoxy)-1-(oxolane-3-carbonyl)piperidine-4-carboxylic acid
3-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyridine
2-(4-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]piperidin-1-yl}phenyl)-1-(pyrrolidin-1-yl)ethan-1-one
5-(propan-2-yl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-(1,3-benzothiazol-2-yl)-N-cyclopropylpiperazine-2-carboxamide