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2-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-N-(2-phenylethyl)acetamide
N-(3,4-difluorophenyl)-1-(pyridin-3-ylmethyl)piperidin-3-amine
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3-(1H-pyrazol-1-yl)benzamide
(4aS,8aS)-2-[2-(1H-1,3-benzodiazol-1-yl)propyl]-decahydroisoquinoline
3-(2-fluorophenyl)-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidine
N,1-dimethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-(4-fluorophenyl)urea
3-{[(5-hydroxypentyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-(1,2,3,4-tetrahydronaphthalen-2-yl)-4-(1H-1,2,4-triazole-5-carbonyl)piperazine
4-(5-{[({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)amino]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
1-[2-({4-cyclopropyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-4-methoxyphenyl]-1H-pyrazole
3-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)-N-propyl-N-(pyridin-3-ylmethyl)propanamide
N-[2-(dimethylamino)ethyl]-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
2-(2-{4-[(2-methyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
3-(3-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}propyl)pyridine
1-(5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)piperazine
N-(2-hydroxyethyl)-5-(methoxymethyl)-N-(1,3-thiazol-2-ylmethyl)thiophene-2-carboxamide
ethyl 2-({5-[(2S,4R,6S)-4-acetamido-6-ethyloxan-2-yl]pyrimidin-2-yl}amino)acetate
1-[4-(2-methylphenoxy)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
4-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-(furan-2-ylmethyl)piperidine
1-{4-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidine-1-carbonyl]phenyl}ethan-1-one
2-(2,3-difluorophenyl)-1-[3-(pyridin-4-yl)azetidin-1-yl]ethan-1-one
(3S,5S)-1-(2,3-dihydro-1H-inden-2-yl)-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
1-[2-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)pyridine-4-carbonyl]-4-methylpiperazine
6-(3-fluoro-4-methylphenyl)-N,N-dimethylpyrazine-2-carboxamide
2,5-dimethyl-3-(4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine
[(4-chlorophenyl)methyl](ethyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
8-(1-ethyl-1H-pyrazole-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl 1-benzyl-5-[(3-methylbutyl)amino]-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylphenyl)methyl]acetamide
4-[({2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)methyl]benzene-1-sulfonamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[(1s,4s)-4-aminocyclohexyl]acetamide
1-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-1H-indole
5-(morpholin-4-ylmethyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}furan-3-carboxamide
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[(1-methylpiperidin-4-yl)methyl]piperazine
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-chloro-4-hydroxyphenyl)ethan-1-one
2-butyl-8-(5-hydroxypyrazine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-1-(2-methoxyethyl)-4-phenylpyrrolidin-3-yl]pyrrolidine-1-sulfonamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
N-cyclopentyl-2-{[2-(2,3-dimethoxyphenyl)ethyl]amino}propanamide
N-({3-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}methyl)propanamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(3-fluoropropyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-(azepan-1-yl)-N-methyl-N-(pyridin-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-cyclohexyl-3-({[(3-methoxyphenyl)methyl]amino}methyl)-N-methylpyridin-2-amine
2-(butylsulfanyl)-5-[1-(pyridin-3-yl)-1H-imidazol-2-yl]pyrimidine
4-{[5-(1-methanesulfonylpyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-propylpiperidine
4-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-1-(3,5-dimethylphenyl)piperazin-2-one
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(2,3-dimethylphenyl)methyl]propanamide
5-methanesulfonyl-N,2-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]pyrimidin-4-amine