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2-amino-6-(4-fluorophenyl)-4-[3-(2-hydroxyethoxy)phenyl]pyridine-3-carbonitrile
1-benzyl-5-(2-methoxypyridine-3-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 2-[1-(3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-3-oxopiperazin-2-yl]acetate
2-phenoxy-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
1-(4-chloro-3-methyl-1H-pyrazole-5-carbonyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
4-chloro-1-methyl-N-[3-(pyridin-3-yloxy)propyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
4-(1-methyl-1H-imidazol-2-yl)-1-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-1H-1,2,3-triazole
2-(3-methyl-5-{2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazol-5-yl}-1H-1,2,4-triazol-1-yl)acetic acid
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-(pyridin-3-yloxy)ethan-1-one
8-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-(4-chlorophenoxy)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]piperidine-4-carboxamide
4-ethyl-5-{[2-(2-fluorophenyl)-1H-imidazol-1-yl]methyl}-2-methyl-1,3-thiazole
N-[2-(azepan-1-yl)ethyl]-N-ethyl-3-(N-methylmethanesulfonamido)propanamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(methylsulfanyl)propan-1-one
7-(2,3-dimethoxyphenyl)-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-[(3,4-difluorophenyl)methyl]-N,N-dimethyl-6-oxo-2,7-diazaspiro[4.5]decane-2-sulfonamide
N-cyclopentyl-4-(4-methanesulfonylphenyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[1-cyclopentyl-4-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
4-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}piperidine
4-[({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)methyl]-1-methyl-1,2,3,4-tetrahydroquinolin-2-one
2-(methylsulfanyl)-N-(propan-2-yl)-N-[(2,4,5-trimethoxyphenyl)methyl]acetamide
1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(propylsulfanyl)ethan-1-one
6-(2,5-dimethylfuran-3-yl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-acetyl-N-(3-{[(2-chlorophenyl)methyl]sulfanyl}propyl)piperidine-3-carboxamide
1-(3-methylbutyl)-8-(pyridin-2-ylmethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 5-{[(3S,5S)-5-(methoxycarbonyl)-1-methylpyrrolidin-3-yl]sulfamoyl}-1-methyl-1H-pyrrole-2-carboxylate
9-(5-ethylthiophene-3-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-5,6-dimethylpyridine-3-carboxamide
4-hydroxy-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(1S,5R)-6-(3-chloro-5-fluorobenzoyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N'1-[(3R,4S)-1-(2-hydroxyethyl)-4-propylpyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
3-[(3R,4S)-1-[2-(3-methylphenyl)acetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
2-(4-methyl-2-{1H-pyrazolo[3,4-b]pyridin-1-yl}phenoxy)acetamide
(1R,2R,6S,7S)-4-(2-methyl-5-propylpyrimidin-4-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
ethyl N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}carbamate
6-[2-(3,4-dimethoxyphenyl)ethyl]-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
2-amino-4-{2-[(propan-2-yl)amino]pyrimidin-5-yl}-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(2S,4R)-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)-1-[(2,4,5-trimethoxyphenyl)methyl]pyrrolidine-2-carboxamide
3-{[5-(4-fluoro-2-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}pyridine
N-(4-methyl-1,3-thiazol-2-yl)-N'-[(2-methylphenyl)methyl]-N'-(prop-2-en-1-yl)ethanediamide
3-[2-(1,3-benzoxazol-2-yl)phenyl]propanamide
4,4-difluoro-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidine
[(3,4-dimethoxyphenyl)methyl]({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amine
1-[4-(difluoromethoxy)-2-methylphenyl]-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
N,5,6-trimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
3-(1H-imidazol-2-yl)-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}benzamide
4-[1-(2H-1,3-benzodioxol-5-yl)-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]thiophene-3-sulfonamide
2-[1-benzyl-5-(5-chloro-2,3-dihydro-1H-indol-2-yl)-1H-1,2,4-triazol-3-yl]acetamide