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2-benzyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1,3-thiazole-4-carboxamide
N-[(2-methoxyphenyl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-(prop-2-en-1-yl)propanamide
N1-[2-(4-methoxyphenyl)phenyl]piperidine-1,3-dicarboxamide
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-(methoxymethyl)furan-2-carboxamide
[(2-chloropyridin-3-yl)methyl](1H-imidazol-2-ylmethyl)methylamine
3-(4-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
3-methyl-N-({1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-3-yl}methyl)but-2-enamide
5-{1-[5-(dimethylcarbamoyl)thiophen-2-yl]-1H-imidazol-2-yl}thiophene-2-carboxylic acid
methyl 3-(4-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
(3R,7S,8aS)-7-{[(2-fluoro-5-methylphenyl)methyl]amino}-3-(2-methylpropyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[1-(2-phenylethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
1-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-phenylethan-1-one
2-methyl-5-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,4-dihydropyridin-4-one
1-[4-(pyridin-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-{2-[1-(2-cyclopropylpyrimidine-5-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
2-methyl-8-[3-(1H-pyrrol-1-yl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(4aS,7aR)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[4-(3-phenylpropyl)-1-[3-(trifluoromethyl)benzenesulfonyl]piperidin-4-yl]methanol
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1,3-thiazol-2-ylmethyl)pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
3-[(2,6-dihydroxyphenyl)formamido]-N-(4-fluoro-2-methylphenyl)propanamide
(1R,5R)-6-(2-methoxyethyl)-3-(5-phenoxyfuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[(4-fluorophenyl)methyl]-1-[(2-methoxyphenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-{[3-methyl-7-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(phenylsulfanyl)acetamide
5-ethyl-N,2-dimethyl-N-[3-(1H-pyrazol-1-yl)propyl]pyrimidin-4-amine
3-(3-fluorophenyl)-4-[3-(1H-pyrazol-1-yl)benzoyl]piperazin-2-one
N-[(4-fluorophenyl)methyl]-3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]propanamide
(2S)-2-[(6-ethyl-2-oxo-1,2-dihydropyridin-4-yl)formamido]-3-(4-hydroxyphenyl)propanamide
3-[2-(2,6-difluorophenyl)ethyl]-1-(5-propyl-1,2-oxazole-4-carbonyl)piperidine
6-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}pyridine-2-carbonitrile
4-{3-cyclopropyl-5-[1-(dimethyl-1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-1,2,4-triazol-1-yl}-3-methylpyridine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-1-[3-(1H-pyrazol-5-yl)phenyl]piperidin-4-amine
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1H-pyrazole-4-carboxamide
(4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}morpholin-3-yl)methanol
4-[4-(1H-pyrazol-4-yl)butanoyl]-1λ6-thiomorpholine-1,1-dione
methyl 2-[(butan-2-yl)sulfamoyl]-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-(oxan-4-yl)piperidine-3-carboxamide
2-(3-methoxypropyl)-9-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-amino-1-(3,4-diethoxybenzoyl)-N-methylpyrrolidine-2-carboxamide
2-{1-[5-(5-methylfuran-2-yl)-1,2,4-triazin-3-yl]piperidin-3-yl}-1H-1,3-benzodiazole
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
4-(2,4-dimethyl-1,4-diazepane-1-carbonyl)-2-(1-ethyl-1H-pyrazol-4-yl)-7-fluoroquinoline
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-(1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
N,N-diethyl-7-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N-(3-methoxypropyl)-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
methyl(2-phenyl-1-{1-[2-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}ethyl)(pyridin-3-ylmethyl)amine
methyl[(3-{2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl](quinolin-8-ylmethyl)amine
1-{[2-methoxy-5-(4-phenyl-1H-imidazol-5-yl)phenyl]methyl}-1H-1,2,4-triazole
N-(2-ethoxyethyl)-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]amine