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2-(4-{1-[2-(4-chlorophenoxy)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)ethan-1-ol
1-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-3,3-diphenylpiperidine
(1R,2R)-2-phenyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropane-1-carboxamide
5-[(4-ethylpiperazin-1-yl)methyl]-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1,2-oxazole-3-carboxamide
6-(2-methoxyphenyl)-N-(oxan-2-ylmethyl)pyridazin-3-amine
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-3-(piperidin-3-yl)benzamide
3-[(4aR,7aS)-4-[2-(methylamino)pyrimidine-5-carbonyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
5-ethyl-1'-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[5-({4-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1-methyl-1H-pyrrol-3-yl]ethan-1-one
1-[2-(4-fluorophenyl)ethyl]-4-[(2-methyl-5-propylpyrimidin-4-yl)amino]pyrrolidin-2-one
2-[(4-methoxyphenyl)methyl]-6-(2,4,5-trimethylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-chloro-2-({4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)-1H-indole
N-(2-chlorophenyl)-2-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-2-oxoacetamide
1,5-dimethyl-3-[3-(morpholin-4-ylmethyl)phenyl]-1H-indazole
3-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-ylmethyl]phenol
[(3-ethoxy-4-methoxyphenyl)methyl]({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
2-(2-fluorophenyl)-4-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-1H-indazole-3-carboxamide
3-ethyl-6-[4-(4-methoxybutyl)piperazine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
2-ethyl-9-[2-hydroxy-2-(4-methoxyphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
2-(2H-1,3-benzodioxol-5-yl)-1-(1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)ethan-1-one
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]benzamide
(2S)-3-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propane-1,2-diol
4,6-dimethyl-2-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyridine-3-carbonitrile
4-(1H-imidazol-2-yl)-1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidine
2-hydroxy-N-[(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]acetamide
2-(furan-2-yl)-N-[(5-methoxy-1H-indol-2-yl)methyl]-2-oxoacetamide
3-methyl-1-(5-methyl-1,3,4-thiadiazol-2-yl)-3-[(2-phenyl-1,3-thiazol-4-yl)methyl]urea
2-[4-(benzyloxy)butanamido]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
1-[(4-methyl-1H-imidazol-2-yl)methyl]-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-(3,4,5-trimethoxyphenyl)ethan-1-one
dimethyl({2-[4-(piperidine-1-carbonyl)phenoxy]phenyl}methyl)amine
8-chloro-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]quinoline-2-carboxamide
2-(pyridin-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide
6,7-dimethoxy-2-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
2-(dimethylamino)-2-(2-methylphenyl)-N-(1,2-oxazol-3-ylmethyl)acetamide
2-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-7-(pyrazin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-methyl-1-{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperidine-3-carboxamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
8-(1H-indol-2-ylmethyl)-1-(2-methoxyethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S)-N3-tert-butyl-N2-(3-methoxyphenyl)-1,2,3,4-tetrahydroisoquinoline-2,3-dicarboxamide
1-[1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(3-methoxyphenoxy)ethan-1-one
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl]propanoate
2-(6-methoxynaphthalen-2-yl)-4-(3-methylpyrazin-2-yl)morpholine
N-{[7-chloro-2-(2,5-dimethoxyphenyl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]furan-2-carboxamide
N-cyclopropyl-4-{methyl[(3-methylpyridin-4-yl)methyl]sulfamoyl}benzamide
1-(cyclohexylmethyl)-6-oxo-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine-3-carboxamide
4-({1-[1-(pyrimidin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)-1,4-diazepan-2-one