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6-{3-oxo-3-[2-(3-phenylpropyl)morpholin-4-yl]propyl}-2,3,4,5-tetrahydropyridazin-3-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(4-methylphenyl)propan-1-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(5-ethylthiophene-3-carbonyl)pyrrolidin-3-yl]methanol
6-{1-[(2-methoxyquinolin-3-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
(3S,9aR)-3-(4-aminobutyl)-8-[(5-methylthiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-2,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,4-dimethyl-3-(2-oxoimidazolidin-1-yl)benzamide
methyl (2S,4R)-1-(cyclohexylmethyl)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
methyl (2R,4S)-4-hydroxy-1-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]piperidine-2-carboxylate
3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]propanamide
2-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N-(propan-2-yl)acetamide
[(5-fluoro-1H-indol-2-yl)methyl](methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
5-cyclopentyl-4-phenyl-1H-imidazole
5-acetyl-N,6-dimethyl-2-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
N-(2-hydroxyethyl)-3-(5-methylthiophen-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
4-(ethylamino)-N-[(2-fluorophenyl)methyl]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(pyridin-4-yl)propan-1-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-oxo-4H-chromene-2-carboxamide
1,4,6-trimethyl-3-{9-methyl-3,9-diazaspiro[5.6]dodecane-3-carbonyl}-1,2-dihydropyridin-2-one
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-3-phenyl-1H-pyrazole-4-carboxamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]ethan-1-one
6-fluoro-2-[({2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}amino)methyl]quinolin-4-ol
1-{1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-4-yl}piperidin-4-ol
{1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-4-yl}methanol
3-phenyl-1-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}pyrrolidin-3-ol
N-methyl-5-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[4-(pyridin-2-yl)butyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
3-[(3-hydroxyazetidin-1-yl)sulfonyl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)benzamide
6-[3-(methoxymethyl)pyrrolidin-1-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4-(oxan-2-ylmethyl)piperidin-4-yl)methanol
2-(methylamino)-1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N,5-dimethyl-N-(quinoxalin-2-ylmethyl)-1,2-oxazole-3-carboxamide
1-(1-{3-benzyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-2-(propan-2-yl)-1H-imidazole
2-(cyclopropylmethyl)-8-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
1-[(4-chloro-3-fluorophenyl)methyl]-4-(oxan-4-yl)piperazine
5-acetyl-6-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
(3S,5R)-N3-[(1-ethylpyrrolidin-2-yl)methyl]-N5-(4-fluorophenyl)-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
3-{[(5-methyl-1,2-oxazol-3-yl)methyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
9-[4-(1H-pyrazol-4-yl)butanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclohexyl-2-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-N-methylacetamide
1-(4-chlorophenyl)-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}cyclopropane-1-carboxamide
4-{[2-(trifluoromethoxy)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
1-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
2-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-4,6-dimethylpyridine-3-carbonitrile
1-(2-chloro-4-fluorobenzoyl)-3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
(3S,4R)-3-methoxy-1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]piperidin-4-amine
N2-benzyl-6-(furan-3-yl)-1,3,5-triazine-2,4-diamine
3-[(3S,4R)-4-(morpholin-4-yl)-1-(pyridin-2-ylmethyl)piperidin-3-yl]-1-(piperidin-1-yl)propan-1-one