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N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
N-benzyl-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
3-(furan-3-ylmethyl)-1-{3-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}urea
({5-[1-(2,1,3-benzoxadiazole-5-carbonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-[5-(propan-2-yl)thiophene-3-carbonyl]-2-(pyrrolidine-1-carbonyl)piperazine
2-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-4,5,6,7-tetrahydro-1,3-benzothiazole
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
methyl 5-[1-(phenylamino)cyclopentanecarbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-methyl-2-[(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)amino]pyridine-4-carboxamide
(3E)-N-(3-chloro-4-propanamidophenyl)-4-phenylbut-3-enamide
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1-(3-phenylphenyl)piperidin-4-amine
(1S,5R)-N-[(3-fluorophenyl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-2-(methylsulfanyl)pyrimidine
1-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
5-(1-{5-[(1E)-1-(furan-2-yl)prop-1-en-2-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)-1H-1,2,3,4-tetrazole
2-{1-[(2-ethoxyphenyl)methyl]-4-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
(2S,4R)-4-amino-1-({2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-N-methylpyrrolidine-2-carboxamide
2-[3-({1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}methyl)phenoxy]acetamide
{2-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]phenyl}methanol
({4-[(dimethylamino)methyl]phenyl}methyl)(methyl){[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
(4aR,7aS)-1-ethyl-4-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(3-hydroxy-3-phenylpropyl)-N,1,4,6-tetramethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{[4-(2-chlorophenyl)-5-[1-(propan-2-yloxy)ethyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-(3-{2,7-diazaspiro[4.5]decan-7-yl}-3-oxopropyl)azepan-2-one
1-(3-ethylpiperazin-1-yl)-3-(2-methylphenoxy)propan-1-one
1-ethyl-8-[(4-hydroxyphenyl)methyl]-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[5-({[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-2-(propan-2-yloxy)phenyl]methanol
2-cyclopropyl-8-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
2-[5-(3,4-dichlorophenoxymethyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
8-{[3-(2-methylphenyl)phenyl]methyl}-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
5-(2-chlorophenyl)-N-{3-[(pyridin-3-yl)amino]propyl}furan-2-carboxamide
N-({7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
1-[(3-acetylphenyl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
2-amino-6-(6-methoxypyridin-3-yl)-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
3-fluoro-5-methyl-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]imidazo[1,2-a]pyridine-2-carboxamide
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-(pyridin-2-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-propylpiperidine
8-fluoro-2-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}quinoline
1-[(4-fluorophenyl)methyl]-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-[2-(piperazin-1-yl)ethyl]-N-[2-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-(8-fluoroquinoline-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
9-[(2-ethoxyphenyl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
3-hydroxy-3-{[(2-hydroxyethyl)amino]methyl}-1-[(3-methoxyphenyl)methyl]piperidin-2-one