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N-[(5-methylpyrazin-2-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-6-oxo-N-(pyridin-3-ylmethyl)-1,6-dihydropyridazine-3-carboxamide
2,6-dimethyl-4-[3-(pyridin-2-yl)azetidine-1-carbonyl]quinoline
N-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylbenzamide
2-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1-benzofuran-7-carboxamide
N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
(3S,4R)-1-(5-acetylthiophene-2-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
ethyl 4-{[1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}piperidine-1-carboxylate
1-[6-(4-methoxyphenyl)-2-(thiomorpholin-4-yl)pyridine-3-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-[(3S,4R)-1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
2-(3,4-dichlorophenyl)-4-[(4,6-dimethylpyrimidin-2-yl)methyl]morpholine
3-(4-hydroxyphenyl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}propan-1-one
(3R,5S)-N3-(4-fluorophenyl)-N5-[(4-methylphenyl)methyl]piperidine-3,5-dicarboxamide
2-[4-(2,5-difluorobenzoyl)morpholin-3-yl]-N-(pyridin-3-ylmethyl)acetamide
4-(1-butyl-1H-imidazol-2-yl)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
4-methyl-2-[1-(1,3-thiazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
N3-cyclooctyl-N5-(1-hydroxy-2-methylpropan-2-yl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-{[1-(2-ethoxypyridine-3-carbonyl)piperidin-4-yl]methyl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-4-(pyrrolidin-3-yl)piperazine
N-ethyl-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-methyl-3-phenyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
1-[(3S,4S)-4-(4-fluorophenyl)-3-hydroxypiperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
3-chloro-N-cyclopentyl-4-[(1-ethylpiperidin-4-yl)oxy]benzamide
(2R,3S,6R)-3-phenyl-5-(pyrazine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-{[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-{[4-(2-hydroxyethoxy)phenyl]methyl}-3-(2-methoxyethyl)piperidine-3-carboxylic acid
4-(4-ethoxy-3-methylphenyl)-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]butanamide
N-methyl-N-(1H-pyrazol-5-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
3-(4-hydroxyphenyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}propanamide
1-methyl-6-propyl-4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-1H-pyrazolo[3,4-d]pyrimidine
5-[2-(dimethylamino)propanoyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(3aR,6aS)-5-{2-[cyclopentyl(methyl)amino]acetyl}-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3-hydroxypropyl)-8-{[3-(methylsulfanyl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-{9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-phenylethan-1-one
2-[2-(dimethylamino)ethyl]-N-(4-fluorophenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-benzyl({1-oxaspiro[4.4]nonan-3-yl}amino)sulfonamide
1-[3-(3-methoxypyrrolidine-1-carbonyl)benzenesulfonyl]-4-methyl-1,4-diazepane
1-[2-(methylsulfanyl)benzoyl]-4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidine
2-methoxy-6-[(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)methyl]phenol
8-(3-methylpyrazin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-benzyl-3-(pyridin-2-ylmethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[4-(3-methylphenyl)phenyl]-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxamide
5-{[(8-methoxyquinolin-5-yl)methyl](methyl)carbamoyl}-1H-imidazole-4-carboxylic acid
N-[2-(1H-imidazol-4-yl)ethyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
8-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(3-fluorophenyl)methyl]-N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-6-oxopiperidine-3-carboxamide
2-(3,5-difluorophenyl)-N-(3,4-dimethyl-1H-pyrazol-5-yl)acetamide
N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amine