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(3aR,7aS)-2-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-(2-methoxy-4-{[methyl(quinoxalin-2-ylmethyl)amino]methyl}phenoxy)propanoic acid
5-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)-1H-1,2,3-benzotriazole
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-methoxyphenyl)methyl]acetamide
4-{[1-(6-aminopyridine-3-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-2-(pyridin-3-yloxy)ethan-1-one
(2R,3R,6R)-5-(cyclopropanesulfonyl)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-({[1-(cyclohex-1-en-1-yl)ethyl]carbamoyl}amino)-2-fluoro-N-methylbenzamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-(2-methylpentanoyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 4-(3-{2-[(5-chloro-2-methoxyphenyl)carbamoyl]ethyl}piperidin-1-yl)piperidine-1-carboxylate
1-(2-amino-6-methyl-1,3-benzothiazol-4-yl)-5-oxopyrrolidine-3-carboxylic acid
methyl({[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl})[1-(pyrimidin-4-yl)ethyl]amine
1-(4-chlorophenyl)-3-cyclopropyl-5-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1H-1,2,4-triazole
2-(3,4-dimethoxyphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
5-[(4-ethylpiperazin-1-yl)methyl]-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2-oxazole-3-carboxamide
N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-3-(prop-2-en-1-yloxy)benzamide
6-oxo-N-(2-phenylethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
N-(1H-imidazol-2-ylmethyl)-2,3-dihydro-1,4-benzodioxine-5-carboxamide
N-(2-methoxyethyl)-5-methyl-4-(methylamino)thieno[2,3-d]pyrimidine-6-carboxamide
1-[2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]pyrrolidin-2-one
N-methyl-3-phenyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
3-[(4-aminopiperidin-1-yl)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
2-[(2-methylnaphthalen-1-yl)methyl]-5-(4-methylpiperazin-1-yl)-2,3-dihydropyridazin-3-one
N'-(2,3-dimethylphenyl)-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}propanediamide
4-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-4-fluoro-N-[(4-methoxyphenyl)methyl]benzamide
N-(4-chloro-2-fluorophenyl)-2-{[(2,3-dimethylphenyl)methyl]amino}acetamide
(2-methoxyethyl)({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})(propan-2-yl)amine
4-(3-benzyl-1,2,4-oxadiazol-5-yl)benzene-1-sulfonamide
2-amino-4-(4-hydroxy-3,5-dimethoxyphenyl)-6-phenylpyridine-3-carbonitrile
1-(3,5-dimethylbenzoyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-(3-fluorophenyl)-3-(1-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
4-benzyl-3-ethyl-1-[2-(2-hydroxyethoxy)ethyl]-1,4-diazepan-5-one
7-chloro-2-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-4H-pyrido[1,2-a]pyrimidin-4-one
1-[4-(4-ethenylbenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-3-phenylpropan-1-ol
N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methyl-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
(2S,4S)-4-amino-1-methyl-N-[3-(4-methylbenzenesulfonamido)propyl]pyrrolidine-2-carboxamide
1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-1H,2H,3H,4H,6H,10bH-pyrimido[2,1-a]isoindol-6-one
N-(1-phenylethyl)-4-{4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-1-yl}benzamide
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]-N-(5-chloro-2-methoxyphenyl)propanamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}methanesulfonamide
N-[2-(3,5-dimethylphenoxy)ethyl]-N-methyl-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
(1R,5R)-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
4-[(2,5-dimethoxyphenyl)methyl]-7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(5-methyl-1,2,4-oxadiazol-3-yl)-1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
4-{2-[1-(2-fluoro-4-methylbenzoyl)piperidin-2-yl]ethyl}morpholine
N-[2-(cyclohex-1-ene-1-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-2-(2-fluorophenyl)acetamide
7-[2-(azepan-1-yl)acetyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[2-amino-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-5-phenylpentan-1-one