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N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-4-(trifluoromethyl)benzamide
3-(dimethylamino)-1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
1-[1-(4-methoxybenzoyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
2-(1H-imidazol-4-yl)-1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)ethan-1-one
2-(azepan-1-yl)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-oxoacetamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,2-oxazole-3-carbonyl)piperidine
(2S)-2-(methoxymethyl)-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}pyrrolidine
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(1H-pyrrole-2-carbonyl)piperidin-4-ol
(3S,4S)-4-(propan-2-yloxy)-1-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-3-ol
4-[({[2-(3-hydroxypiperidin-1-yl)-5,6,7-trimethoxyquinolin-3-yl]methyl}amino)methyl]benzene-1-sulfonamide
1-ethyl-8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S)-4-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-ethyl-3-methylpiperazin-2-one
1-(2-methoxyphenyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-pyrazole-4-carboxamide
2-(4-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-ol
(3S,4S)-1-(5,6-dimethylpyrimidin-4-yl)-4-(naphthalen-2-yl)piperidin-3-ol
N-methyl-N-(oxolan-2-ylmethyl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-{2-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}-2-methylfuran-3-carboxamide
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
methyl 6-(but-2-ynoyl)-2-[(3,5-dimethylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(3-acetylphenyl)-1-(3-methylbut-2-en-1-yl)-6-(5-methylpyrazine-2-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{2-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-3,3-dimethylurea
[(3,5-difluoro-4-methoxyphenyl)methyl](methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
{[(3R,4S)-4-cyclopropyl-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl]sulfamoyl}dimethylamine
2-(5-chloro-2-fluorobenzoyl)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
4-{[(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)amino]methyl}-6-ethyl-2H-chromen-2-one
3-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridine
4-{[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]methyl}benzonitrile
3-(6-methoxypyridin-3-yl)-5-[(pyridin-2-ylmethyl)sulfamoyl]benzoic acid
4-(1H-imidazol-2-yl)-3-methyl-2-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(1S,5R)-6-(cyclobutylmethyl)-3-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-N-[(3-methylphenyl)methyl]pyrimidin-2-amine
N-(4-{[(2H-1,3-benzodioxol-5-ylmethyl)carbamoyl]methyl}phenyl)butanamide
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
2,2-dimethyl-1-(4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperazin-1-yl)propan-1-one
2-{3-[2-(methylsulfanyl)ethyl]-5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]-1H-1,2,4-triazol-1-yl}acetic acid
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-2-(2-oxopyrrolidin-1-yl)acetamide
N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
1-{[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidine-4-carboxamide
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}pyrrolidin-2-one
5-[3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
N-({7-[(3-ethoxy-4-hydroxyphenyl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenoxypropanamide
2-[6-(piperidin-1-yl)pyridin-3-yl]-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]acetic acid
1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
2-(dimethylamino)-7-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 4-{[4-(2-{[(3-chlorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]methyl}benzoate
1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
2-methoxy-3-(3-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine
8-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-methyl-1-benzofuran-5-carboxamide