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6-tert-butyl-2-[3-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
3-(4-fluorophenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
N-(butan-2-yl)-2-(dimethyl-1,3-thiazol-4-yl)-N-(pyridin-4-ylmethyl)acetamide
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-(2-{methyl[(3-methylpyridin-4-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
9-(1,3-benzothiazole-6-carbonyl)-5-methoxy-1-oxa-9-azaspiro[5.5]undecane
2-cyclohexyl-6-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
N-cyclohexyl-2-[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]butanamide
2-methyl-4-{3-[(1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]phenyl}butan-2-ol
2-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
methyl 6-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-3-(5-methylthiophene-2-amido)thieno[2,3-b]pyridine-2-carboxylate
6-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
1-{2-hydroxy-3-[4-methoxy-2-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
6-(morpholine-4-sulfonyl)-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-{[2-(4-methylpyrimidin-2-yl)phenyl]methyl}piperidin-4-one
2-(cyclopent-1-ene-1-carbonyl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
3-[(dimethylamino)methyl]-1-(quinoxaline-5-carbonyl)piperidin-3-ol
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-2-(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)acetamide
5-({5-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-4-phenyl-1H-imidazol-1-yl}methyl)-N-methylfuran-2-carboxamide
2-methyl-4-(4-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}phenyl)but-3-yn-2-ol
6-ethyl-4-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-{4-[2-(phenylsulfanyl)ethyl]piperazin-1-yl}-1-azabicyclo[2.2.2]octane
1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-3-methylbutan-1-ol
N-cyclopropyl-2-(4-fluorophenyl)-N-({4-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)acetamide
2-[5-(3-aminophenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
(2S,4S)-4-amino-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-N-ethylpyrrolidine-2-carboxamide
4-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-{2-[4-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-{5-[(methylsulfanyl)methyl]pyridin-2-yl}pyrrolidin-3-yl]methanol
(1S,5R)-6-benzyl-3-(1H-indol-5-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(3-cyanopiperidin-1-yl)sulfonyl]-N-(2,2,2-trifluoroethyl)benzamide
(7S,9aR)-N-(3-fluorophenyl)-7-(hydroxymethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
2-{[(5-acetylthiophen-2-yl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
2-[4-(2,4-difluorobenzoyl)-2-oxopiperazin-1-yl]benzonitrile
4-benzyl-1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-(4-methylbenzoyl)piperidin-4-amine
1-[2-methoxy-4-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N2,N4,N4,5-tetramethyl-N2-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrimidine-2,4-diamine
(4aR,8aS)-1-[2-(3-fluorophenyl)ethyl]-6-[2-(thiophen-3-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
(3S,5S)-1-[3-(methylsulfanyl)propyl]-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-[2-chloro-5-(morpholine-4-carbonyl)phenyl]-1,4-diazepane-1-carboxamide
N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1-(pyridine-4-carbonyl)piperidin-4-amine
methyl({[5-(pyridin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl})(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
1-(3-methylbutyl)-8-(oxan-4-yl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[6-oxo-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]cyclopropane-1-carboxamide
N-(1H-imidazol-2-ylmethyl)-4-(piperazine-1-sulfonyl)benzamide
ethyl 2-chloro-5-({[2-(N-methylmethanesulfonamido)ethyl]carbamoyl}amino)benzoate
2-{4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N-(2-methyl-1-benzofuran-7-yl)acetamide
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide