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1-cycloheptyl-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
1-({4-methyl-5-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
1-{[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-4-ol
{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}[2-(3-methoxyphenyl)ethyl]amine
8-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(cyclopropylmethyl)({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})propylamine
1-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-4-phenoxypiperidine-4-carboxylic acid
2-{2-oxo-2-[4-(2-oxo-1,3-oxazolidin-3-yl)piperidin-1-yl]ethyl}-2,3-dihydro-1,2-benzothiazol-3-one
N-{1-[(4-fluorophenyl)methyl]-7-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
(4aS,7aR)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{3-[(2-fluoroethyl)carbamoyl]benzenesulfonyl}-N-methylpiperidine-2-carboxamide
N-[3-(2-fluorophenyl)propyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-(3-{6-[(propan-2-yl)amino]pyrimidin-4-yl}phenyl)ethan-1-one
ethyl 3-[(3-chlorophenyl)methyl]-1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidine-3-carboxylate
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-3-carboxylic acid
N1,N1,N4-trimethyl-N4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-1,4-dicarboxamide
6-chloro-N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2H-chromene-3-carboxamide
6-fluoro-3-[2-(1-methylpiperidin-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
2-methyl-4-[4-({4-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}methyl)phenyl]butan-2-ol
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2-oxoimidazolidine-4-carboxamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-methoxypropan-1-one
5-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-2-(pyridin-3-yl)pyrimidin-4-ol
1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[1-(1-methyl-1H-pyrazol-5-yl)propyl]urea
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(trifluoromethyl)phenyl]urea
(1S,4S)-2-(2-chlorophenyl)-5-(quinoxalin-5-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
4-(propylsulfamoyl)-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
methyl (2S)-2-{[2-(2-methylbenzamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-5-yl]formamido}-2-phenylacetate
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-1-methyl-1H-imidazole-2-carboxamide
4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}morpholine
4-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoacetamide
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[(4-ethylphenyl)methyl]methylamine
4-(5-chloro-2-methoxyphenyl)-3-[(propan-2-yloxy)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-benzyl-4-(4-chloro-3-fluorobenzoyl)piperazin-2-one
N-{[4-(dimethylsulfamoyl)phenyl]methyl}-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
2-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-2-oxo-N-(propan-2-yl)acetamide
7-(cyclopropylmethyl)-2-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
3-(4-methylpiperazine-1-carbonyl)-N-(2-methylpropyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]methyl}-2,1,3-benzoxadiazole
6-(4-chlorophenyl)-N-[2-(1H-pyrazol-1-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-ethyl-1'-(3-phenyl-1,2,4-oxadiazol-5-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-2,1,3-benzothiadiazole
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[(3-fluoro-4-methylphenyl)methyl]benzamide
methyl 2-{[(3-chlorophenyl)methyl]sulfamoyl}-6-[(2E)-4-methylpent-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{1-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1H-imidazol-2-yl}-2-ethoxyphenol
4-[(3-methoxyphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-N-ethylpyrimidin-2-amine
1-(oxolan-2-ylmethyl)-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
3-{[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine