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N-(3-methylphenyl)-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carboxamide
3-{imidazo[1,2-a]pyridin-2-ylmethyl}-3,4-dihydroquinazolin-4-one
11-(ethylamino)-4-[2-(3-fluorophenyl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(1S,5R)-6-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-7-fluoro-2-methylquinoline-4-carboxamide
3-benzyl-5-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazol-5-yl]-1H-1,2,4-triazole
2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-phenylpropanamide
2-{4-cycloheptyl-1-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
4-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-1-ethylpyrrolidin-2-one
1-(1H-imidazol-2-ylmethyl)-4-(3-methylpyridin-4-yl)piperazine
1-(2-amino-9H-purin-6-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(dimethyl-1,2-oxazole-4-carbonyl)-N-(3,4-dimethylphenyl)piperidin-3-amine
N-[(6-chloropyridin-3-yl)methyl]-2-(dimethylamino)-2-(4-fluorophenyl)-N-methylacetamide
1-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1H,4H,6H,7H-pyrano[4,3-c]pyrazole-3-carboxamide
N-ethyl-5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]pyrimidin-2-amine
6-(2-aminoethyl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)pyrimidin-4-amine
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[(4-cyanophenyl)methyl]propanamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,3,5-trimethyl-1H-pyrazole-4-sulfonamide
ethyl 1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
(3R,5R)-N-[2-(pyridin-2-ylsulfanyl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
3-[2-(4-chlorophenyl)morpholine-4-carbonyl]-6-ethyl-1,5-dimethyl-1,2-dihydropyridin-2-one
3-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
4-{4-ethyl-6-[3-(morpholin-4-yl)piperidin-1-yl]pyrimidin-2-yl}morpholine
4-ethyl-3-({1-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 5-cyclopentanecarbonyl-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylate
3-(3-hydroxy-3-methylbutyl)-N-(1-methyl-6-oxopiperidin-3-yl)benzamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(3-chlorophenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3E)-2-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]hept-3-enoic acid
N-(2-hydroxyethyl)-2,6-dimethyl-N-[(5-methylthiophen-2-yl)methyl]pyridine-4-carboxamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-methyl-1H-pyrazole-5-carboxamide
4-(3-fluorophenoxy)-1-(4-methylpyrimidine-5-carbonyl)piperidine-4-carboxylic acid
4-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]benzonitrile
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-5-methylthieno[2,3-d]pyrimidin-4-amine
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
2-(3-fluorophenoxy)-1-{4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
N-[cyclopropyl(pyridin-2-yl)methyl]-6-ethyl-N,2-dimethylquinoline-4-carboxamide
2-ethyl-5-(2-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-6-methyl-3,4-dihydropyrimidin-4-one
4-(dimethyl-1,3-thiazole-5-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
1-({1-[2-(4-methoxyphenoxy)ethyl]pyrrolidin-2-yl}methyl)-1H-pyrazole
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
4-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
N,1-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-4-methylpiperazin-2-one
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-cyclopropyl-N-ethylpropanamide
3-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(1,3-benzoxazol-2-ylmethyl)methylamine
N-[2-(dimethylsulfamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-4-carboxamide
N,N-dimethyl-5-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)pyrrolidin-2-yl]thiophene-2-carboxamide