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1-cyclopentyl-6-oxo-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide
4-[4-(naphthalen-1-yl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidine
[(4-cyclopropyl-5-{1-[(4-fluoro-3-methylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(morpholin-4-yl)ethan-1-one
2-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-[1-(pyridin-2-yl)propan-2-yl]acetamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}acetamide
4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1-(2-methylphenyl)piperazin-2-one
2-{2-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinolin-1-yl}acetic acid
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N,5-dimethyl-N-(1,2-oxazol-3-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
5-acetyl-6-methyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(5-methylthiophen-2-yl)methyl]-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-[2-(pyrrolidin-1-yl)ethyl]pyrimidin-2-amine
2-(4-{[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]sulfonyl}phenoxy)acetamide
4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholine
[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
N-ethyl-1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)pyrrolidine-3-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-3-[ethyl(pyridin-4-ylmethyl)amino]piperidine-1-carboxamide
[(2S,6S)-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
4-(4-chlorophenyl)-3-[(methylamino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-2-ethoxypyridine
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(pyrazine-2-carbonyl)piperidine-4-carboxylic acid
2-(dimethylamino)-2-(4-methylphenyl)-N-(quinolin-4-ylmethyl)acetamide
2-methoxy-4-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,5,7-trimethyl-1H-indole-2-carboxamide
1-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine-4-carboxamide
(3S)-2-(5-propyl-1,2-oxazole-3-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-3-carboxylic acid
(2S)-N2-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}pyrrolidine-1,2-dicarboxamide
(3S,4R)-1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-4-methylpiperidine-3,4-diol
3-{1-[(5-methyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}benzoic acid
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
5-(4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
9-(furan-3-ylmethyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(pyridin-2-ylmethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
{4-[2,4-dichloro-3-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}methanamine
1-(2-methoxyphenyl)-4-[(3-methoxypyrrolidin-1-yl)methyl]-1H-pyrazole
2-ethoxy-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
3-hexyl-8-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-benzyl-3-{[1-(1-methoxypropan-2-yl)piperidin-4-yl]oxy}benzamide
(3S,4R)-1-(2-methoxyacetyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
5-methoxy-4-oxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,4-dihydropyridine-2-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]benzamide
2-(8-{[4-(furan-2-yl)phenyl]methyl}-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl)acetamide
4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]piperidine
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]amino}-N-methylpyrrolidine-2-carboxamide
11-{[(2-fluorophenyl)methyl]amino}-4-[2-(morpholin-4-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[1-(cyclohexylmethyl)-4-(quinolin-8-ylmethyl)piperazin-2-yl]ethan-1-ol