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1-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-4-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]butan-1-one
3-[2-(4-aminoazepan-1-yl)-2-oxoethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
1-(2-chloroprop-2-en-1-yl)-7-fluoro-3-({[3-(morpholin-4-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
5-[2-(4-methoxyphenyl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(hydroxymethyl)azepan-4-ol
4-phenyl-1-(prop-2-yn-1-yl)-5-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
N-methyl-N-(oxan-2-ylmethyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-{5-[1-(1,3-benzothiazol-2-ylmethyl)-1H-imidazol-2-yl]thiophen-2-yl}prop-2-yn-1-ol
1-cyclopentyl-5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-N-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[2-(oxan-2-yl)ethyl]propanamide
N-[3-oxo-3-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propyl]acetamide
N-(3-ethoxypropyl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
2-(4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-1,3-benzoxazole
(1S,5R)-3-cyclopentyl-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}acetic acid
6-methoxy-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-4-amine
1-{2-[({2-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]phenyl}methyl)amino]ethyl}pyrrolidin-2-one
2-amino-4-({[(1R,2R)-2-hydroxycyclohexyl]methyl}amino)quinazoline-6-carboxylic acid
5-{[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
2-cyclopropyl-9-(2,6-dimethoxypyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(6-methylpyridin-2-yl)methyl]-5-(propan-2-yl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-fluoro-N-({3-methyl-7-[(3-methylquinoxalin-2-yl)methyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)benzamide
6,8-dimethyl-3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
1-[1-(cyclohexylmethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
N,N-dimethyl-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazine-1-sulfonamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(2-methylpyrimidin-4-yl)-decahydro-1,6-naphthyridin-2-one
9-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-1,4,9-triazaspiro[5.5]undecan-5-one
N-[(2R)-1-[3-(2-ethylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]-1-oxobutan-2-yl]acetamide
4-({[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl](methyl)amino}methyl)-1-ethylpyrrolidin-2-one
3-[(4-{[1-(morpholin-4-yl)propan-2-yl]amino}piperidin-1-yl)methyl]phenol
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
2-(3,4-dimethylphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
(2R,3R,6R)-3-(4-methylphenyl)-5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-3-ethoxypropan-1-one
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]cyclohexanecarboxamide
4-[(3-methoxypropyl)amino]-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
1-(pyridin-3-ylmethyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
3-({4-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}methyl)-3,4-dihydroquinazolin-4-one
(3R,4R)-3,4-dimethyl-1-{[4-(morpholine-4-sulfonyl)phenyl]methyl}pyrrolidin-3-ol
3-{[(5-methyl-1,2-oxazol-3-yl)formamido]methyl}-N-(4-phenoxyphenyl)piperidine-1-carboxamide
(1R,3S)-7-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-ethoxy-7-azaspiro[3.5]nonan-1-ol
3-[(diethylamino)methyl]-N-(2,3-dihydro-1,4-benzodioxin-6-yl)benzamide
6-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}pyridine-3-carbonitrile
(3R,4R)-1-(2-aminopyrimidin-4-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
3-{1-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-1H-1,3-benzodiazol-2-yl}propan-1-ol
4-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]benzene-1-sulfonamide
1-methyl-4-(3,3,4,4-tetrafluorobutyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(3-methoxyphenyl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(3-methoxyphenyl)propan-1-one