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6-[(diethylamino)methyl]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
5-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-[furan-2-yl(phenyl)methyl]propanamide
N,5-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(1,4-dioxan-2-ylmethyl)-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
N-[(2R,3R)-1'-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
2-{5-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-2-(1H-1,2,4-triazol-3-yl)benzamide
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
2-(isoquinolin-5-yl)pyridine-3-carboxamide
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
(3aS,6aR)-5-(6-methoxypyrimidin-4-yl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
7-fluoro-4-[4-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}benzamide
3-[(2-methylphenyl)methyl]-3,4-dihydropteridin-4-one
N-methyl-4-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(2S)-4-(methylsulfanyl)-2-[4-(3-methylthiophen-2-yl)-1H-1,2,3-triazol-1-yl]butanoic acid
5-cyclopropanecarbonyl-1'-(1-ethyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-amino-1-{[4-(methylsulfamoyl)phenyl]methyl}pyrrolidine-3-carboxylic acid
1-[3-(2-fluorophenyl)propanoyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
3-(1H-1,3-benzodiazol-1-yl)-1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
1,3-dimethyl-2,6-dioxo-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[(2R)-1-hydroxy-3-methylbutan-2-yl]-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(2S,4R)-4-amino-1-(2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
N-[2-(2-fluorophenoxy)ethyl]-4-(1H-pyrazol-4-yl)butanamide
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-[(3-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
3-(4-fluorophenyl)-4-[4-(1H-imidazol-1-yl)benzoyl]piperazin-2-one
1-(2-phenoxyethyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
ethyl 4-[3-(3-chlorobenzoyl)piperidin-1-yl]piperidine-1-carboxylate
8-[2-(1H-imidazol-1-yl)acetyl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-(dimethylamino)-2-(2-methylphenyl)ethan-1-one
8-(4-chloro-3-fluorobenzoyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(3S,9aR)-8-[(3-fluorophenyl)methyl]-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3S,4R)-4-(2-methylphenyl)-1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]pyrrolidine-3-carboxylic acid
3-(3-oxo-4-phenylpiperazine-1-carbonyl)benzonitrile
N-benzyl-5-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}pyrimidin-2-amine
N-[3-methyl-1-(pyridin-3-yl)butyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[2-(1H-indol-3-yl)ethyl]-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
1-[6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridazin-3-yl]azepane
N-[2-(2-methylpropanesulfonyl)ethyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
(2S)-2-[(2,3,5,6-tetramethylphenyl)formamido]propanamide
N-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-1,2,5-thiadiazole-3-carboxamide
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-2-(pyridin-3-yl)quinoline
3-chloro-N-[(1R,3S)-3-[(furan-3-ylmethyl)(methyl)carbamoyl]cyclopentyl]thiophene-2-carboxamide
4-methoxy-N-{1-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide