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N-[2-(2-chlorophenyl)ethyl]-1-[(4-chlorophenyl)methyl]-6-oxopiperidine-3-carboxamide
2-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]pyridine-3-carbonitrile
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidine
5-{2-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(2-methoxyphenoxy)-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)acetamide
N-[(1S,2R)-2-aminocyclobutyl]-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
(2S)-2-hydroxy-1-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-phenylethan-1-one
1-{2,4-dimethyl-6-[1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}-1H-pyrazole
N-(oxan-3-ylmethyl)-2-(3-phenylpiperidin-1-yl)acetamide
methyl (2S,4R)-4-(4-chloro-2-propanamidobenzamido)-1-methylpyrrolidine-2-carboxylate
2-(5-methyl-1,2-oxazole-3-carbonyl)-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-yl)acetic acid
1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
2-({2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}sulfanyl)-6-methyl-3,4-dihydropyrimidin-4-one
methyl({[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl})[(4-methylphenyl)methyl]amine
1-[6-(dimethylcarbamoyl)pyrazin-2-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(2-methylpropyl)({[5-(oxolan-2-yl)thiophen-2-yl]methyl})(pyridin-2-ylmethyl)amine
2-{[3-(cyclohexylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3-methyl-3H-imidazo[4,5-b]pyridine
1-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
(2E)-N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-3-(4-methoxyphenyl)prop-2-enamide
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-4-methyl-1H-imidazole-5-carboxamide
N-[3-(1H-pyrazol-5-yl)phenyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine-4-carboxamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-(pyridine-4-carbonyl)piperidin-4-ol
(4aR,7aS)-1-(3-methylbut-2-en-1-yl)-4-[2-(phenylsulfanyl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]benzamide
2-(2-{[methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amino]methyl}phenoxy)propanoic acid
5-ethyl-N,2-dimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]pyrimidin-4-amine
4-[(2-butyl-4-methyl-3-oxopiperazin-1-yl)sulfonyl]-N-methylthiophene-2-carboxamide
[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
dimethyl({[2-(3,4,5-trimethoxyphenoxy)phenyl]methyl})amine
(4aS,8aR)-1-(3-methoxypropyl)-6-(1,3-oxazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
ethyl 1-[2-(4-methoxyphenyl)ethyl]-5-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{5-[2-(2-methylphenyl)ethyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl}butan-2-ol
5-chloro-2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
1-methyl-5-[3-(2,2,2-trifluoroethoxy)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
(3R,4S)-1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3,4-dimethylpiperidin-4-ol
(2R,6R)-4-(3-methanesulfonamidopropanoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1'-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
(1S,5R)-6-[5-(4-chloro-2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
2-oxo-N-[2-(propylsulfanyl)ethyl]-1,2-dihydroquinoline-4-carboxamide
4-[(3-carboxy-4-methoxyphenyl)methyl]-1-methylpiperazine-2-carboxylic acid
(2R,3R,6R)-5-(1H-indole-7-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-amino-6-(2-fluorophenyl)-4-(furan-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(4-methoxyphenyl)methyl]-3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]propanamide
2-hydroxy-N-({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}methyl)acetamide
N-(1-benzylpyrrolidin-3-yl)-3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}propanamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2,6-dimethylquinoline-3-carboxamide