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1-(5-{[benzyl(methyl)amino]methyl}-2-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
(4aS,8aR)-6-(oxan-4-yl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
ethyl 5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(4aR,6R,8aS)-8a-(methoxymethyl)-2-(4-methylpyridin-2-yl)-6-(morpholin-4-yl)-decahydroisoquinoline
N-(2H-1,3-benzodioxol-5-yl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
3-{[(5-ethylpyrimidin-2-yl)amino]methyl}-2-methoxy-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-(piperidin-3-ylmethyl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-6-(4-chloro-2-methylbenzoyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)carbamoyl]pyridin-1-ium-1-olate
3-cyclopropyl-6-[3-(4-fluorophenyl)propyl]-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
2-(cyclopropylmethyl)-1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-{3-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]phenoxy}acetamide
(1S,5R)-3-[2-(benzyloxy)acetyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[4-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperazin-1-yl]-1-(pyrrolidin-1-yl)ethan-1-one
3-[2-(3,4-difluorophenyl)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
{4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]morpholin-3-yl}methanol
3-(3-hydroxyquinoxalin-2-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylpropanamide
1-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-4-(pyrrolidin-1-yl)piperidine
N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-N-cyclopentyl-2-methoxybenzamide
(1S,6R)-N-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
3-{2-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-(cyclopropylmethyl)-1,4-diazepan-5-one
2-(1-hydroxypropyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl 4-({3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)benzoate
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-1,2-oxazole-3-carboxamide
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylsulfanyl)ethan-1-one
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[(cyclopropylmethyl)sulfanyl]ethan-1-one
14-(3,5-difluoro-4-methoxyphenyl)-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-{3-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-(1,2-oxazol-3-ylmethyl)pyrimidin-2-amine
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-7-fluoro-2-methylquinoline
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(morpholin-2-yl)ethan-1-one
1-(5-chlorofuran-2-carbonyl)-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
methyl (2R,4S)-4-hydroxy-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperidine-2-carboxylate
3-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}piperidin-3-ol
(3S,5R)-1-(1-propyl-1H-pyrazole-5-carbonyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]-1,2,3-thiadiazole-4-carboxamide
1-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-3-(hydroxymethyl)piperidin-3-ol
(4aS,8aR)-1-(3-hydroxypropyl)-6-{pyrazolo[1,5-a]pyridine-2-carbonyl}-decahydro-1,6-naphthyridin-2-one
4-methyl-1-{[3-(methylsulfanyl)phenyl]methyl}piperidine-4-carbonitrile
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-[3-(propoxymethyl)pyrrolidin-1-yl]propan-1-one
3-(1H-1,3-benzodiazol-2-yl)-N-methyl-N-(quinolin-6-ylmethyl)propanamide
N-ethyl-5-({4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidin-2-amine
(1S,5R)-6-benzyl-3-(6-methylpyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(2-methyl-2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-4-yl]methanesulfonamide
2-cyclopropyl-N-[(2,3-difluorophenyl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-hydroxy-N,N-bis(2-hydroxyethyl)-2-phenylpyrimidine-5-carboxamide
methyl 3-ethyl-2-[(E)-2-phenylethenyl]-3H-imidazo[4,5-b]pyridine-6-carboxylate
2-[(5-methylpyrazin-2-yl)methyl]-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1-methyl-1,2-dihydropyridin-2-one