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3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)piperidine
8-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-[({[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}amino)methyl]piperidin-3-ol
5-acetyl-2,4-dimethyl-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-pyrrole-3-carboxamide
3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-7-chloroquinolin-4-ol
4-hydroxy-N-[2-(propylsulfanyl)phenyl]-4-(pyridin-3-yl)piperidine-1-carboxamide
5-{[2-(4-fluorophenyl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-ethyl-N-[2-(3-fluorophenyl)ethyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
3-(4-fluorophenyl)-3-{imidazo[2,1-b][1,3]thiazol-6-ylformamido}propanoic acid
7-(2-methoxyethyl)-2-(5-propyl-1,3,4-thiadiazol-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(pyridin-3-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
4-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidine
ethyl 5-[(2S,4R,6R)-4-acetamido-6-phenyloxan-2-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]oxolane-3-carboxamide
(3aR,6aR)-2-methanesulfonyl-5-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3R,4S)-4-(4-methoxyphenyl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)pyrrolidin-3-amine
{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]({5-[1-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-pyrazol-3-yl]furan-2-yl}methyl)amine
1-(cyclopropylmethyl)-4-(6-ethyl-2-methylpyrimidin-4-yl)-2-(propan-2-yl)-1,4-diazepane
1-[4-(furan-2-yl)pyrimidin-2-yl]-N-[(3-methoxyphenyl)methyl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]-1-methyl-1H-indole-6-carboxamide
4-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(propan-2-yl)pyrimidine
1-({2-[2-(dimethylamino)ethoxy]phenyl}methyl)-N,N-dimethylpyrrolidin-3-amine
N-cyclohexyl-3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propanamide
1-(2-phenylethyl)-N-[(4-phenyloxan-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
6-[1-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)piperidin-4-yl]pyrimidin-4-ol
8-(2-phenylpropyl)-2-(pyridin-3-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
8-chloro-2-[4-(1-ethylpiperidin-4-yl)piperazin-1-yl]quinoline
2-(ethylamino)-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]pyrimidine-5-carboxamide
N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(3-chlorophenyl)-1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-3-phenylpropan-1-one
1-[(5-ethylfuran-2-yl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
6-(2-aminoethyl)-N,2-dimethyl-N-[1-(pyrimidin-4-yl)ethyl]pyrimidin-4-amine
1-[(2,4-dimethylphenyl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2,2-diphenylacetamide
(1R,5R)-3-(2,4-difluorobenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
8-methyl-3-[(4-methyl-1H-imidazol-2-yl)methyl]-3,4-dihydroquinazolin-4-one
N-cyclopropyl-2-[4-({[(3-methyloxetan-3-yl)methyl]carbamoyl}amino)phenyl]acetamide
(1-{[4-(2,1,3-benzothiadiazol-5-yl)-1H-1,2,3-triazol-1-yl]methyl}cyclopropyl)methanol
N2-{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}-N4,N4,5-trimethylpyrimidine-2,4-diamine
6-{4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butanoyl}-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
5-[(3-fluorophenyl)methyl]-7-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
5-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
4-(2-chlorophenyl)-6-(1H-pyrazol-1-yl)pyrimidine
N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)pent-4-enamide
3-{[2-(2-chlorophenyl)-2-hydroxyethyl]amino}-N-(2-methylphenyl)propanamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-methyl-1,3-oxazole-5-carboxamide