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2-{1-[(4-ethoxyphenyl)methyl]-4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(morpholin-4-yl)-1-(4-phenyl-1,4-diazepan-1-yl)-2-(pyridin-3-yl)ethan-1-one
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)cyclohexanecarboxamide
5-(4-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-1H-indole
1-[2-(cyclopent-2-en-1-yl)acetyl]-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
1-(4-fluoro-2-methylphenyl)-3-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}urea
1-[(2-fluoro-4-methoxyphenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
3-[(4-cyclopentyl-3-oxopiperazin-1-yl)methyl]-7-methoxy-1,2-dihydroquinolin-2-one
ethyl 4-(cyclopropylmethyl)-1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidine-4-carboxylate
2-({dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)-1-[3-(trifluoromethyl)phenyl]ethan-1-ol
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1H-indene-5-carboxamide
1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-propoxyethan-1-one
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[3-(1H-imidazol-1-yl)propyl]acetamide
3-[3-cyclopropyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]quinoline
3-(1-{[5-(3-chlorophenyl)furan-2-yl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
N-methyl-2-oxo-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]propanamide
N2-cyclopropyl-N4-[3-(pyridin-3-yloxy)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
5-{2-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(5-phenyl-4H-1,2,4-triazol-3-yl)-1-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
6-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
6-(1,4-dioxan-2-yl)-3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
4-{[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-methyl-1H-pyrazole
3-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)benzonitrile
4-cyclopropanecarbonyl-N-[3-fluoro-4-(trifluoromethyl)phenyl]-1,4-diazepane-1-carboxamide
N-cyclopropyl-1-{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
(1S,5R)-6-benzyl-3-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
N-{[4-(oxolan-3-yloxy)phenyl]methyl}-4-phenyl-N-(pyridin-2-ylmethyl)benzamide
(3S,4R)-4-methyl-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3,4-diol
1-{4-[(2-hydroxy-2-phenylethyl)(methyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
1-cyclopentyl-N3-ethyl-4-oxo-N5-{[3-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
2-amino-8-(2-methoxyquinolin-3-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-5-(methoxymethyl)-N-methyl-1,3,4-oxadiazole-2-carboxamide
N-(2-oxo-2-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}ethyl)benzamide
3-{4-phenyl-5-[(1E)-1-phenylprop-1-en-2-yl]-1H-imidazol-1-yl}-1λ6-thiolane-1,1-dione
butyl(methyl){[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}amine
3-[(2-aminopyridin-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}-N,N-dimethylpyrimidin-2-amine
N-[2-(2-chlorophenyl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1,9-dioxaspiro[5.5]undecan-4-amine
1-ethyl-3-methyl-8-(3-phenylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-benzyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-4-phenylpiperidine
4-(2-methylphenoxy)-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidine
3-(3-methylcinnolin-5-yl)-1-[1-(morpholin-4-ylmethyl)cyclohexyl]urea
8-(4-carboxy-1,3-oxazol-2-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 6-[(2,5-dimethylphenyl)methyl]-2-[(1-methoxypropan-2-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3aS,6aS)-2-(cyclopentylmethyl)-5-(3-methoxypropanoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-4-(4-{[4-(4-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl}phenyl)butan-2-ol