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[1-(2,3-dihydro-1H-inden-2-yl)-3-[(2-fluorophenyl)methyl]piperidin-3-yl]methanol
5-cyclopropyl-N-ethyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carboxamide
2-chloro-5-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrazine
3-hexyl-8-(oxolan-3-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(2-ethyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-(1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
1'-[(3-methyl-1,2-oxazol-5-yl)methyl]spiro[indene-1,4'-piperidine]
2-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
7-(2-methoxypyridine-3-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-methyl-3-[(pyridin-3-ylmethyl)amino]benzamide
(1R,5S)-3-{[1-(3-methylbutyl)-1H-1,3-benzodiazol-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
N-{4-[2-amino-3-cyano-6-(3-methoxyphenyl)pyridin-4-yl]phenyl}acetamide
N-cyclohexyl-3-propyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
3-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-[3-(propan-2-yloxy)phenyl]urea
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]({[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl})ethylamine
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[4-(2-methylphenyl)benzoyl]pyrrolidin-3-yl]methanol
N-(2-ethyl-1,3-dihydroxypropan-2-yl)-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
4-{[5-(1-cyclohexylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(3,4-difluorophenyl)methyl]piperidine
3-(pyridin-2-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propan-1-one
N-cyclohexyl-3-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)amino]propanamide
5-(phenoxymethyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-3-carboxamide
2-(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(2-phenylphenyl)methyl]pyrimidin-2-amine
2-(dimethylamino)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-(3-methylphenyl)acetamide
4-(2,1,3-benzoxadiazole-5-carbonyl)-1-[(3-methylphenyl)methyl]piperazin-2-one
N,N-diethyl-1-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}pyrrolidin-3-amine
3-{4-[(2,3-dihydroxypropyl)(methyl)amino]pyrimidin-2-yl}benzoic acid
1-[2-(2-oxopyrrolidin-1-yl)ethyl]-5,5-diphenylpiperidin-2-one
ethyl 1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-4-(2-phenylethyl)piperidine-4-carboxylate
N-methyl-2-(pyridin-3-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-5-carboxamide
2-(methoxymethyl)-5-(oxan-2-ylmethyl)-1,3-benzoxazole
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl][(1-methyl-1H-imidazol-2-yl)methyl]amine
methyl 6-(5-chloro-3-methyl-1H-indole-2-carbonyl)-2-(ethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-methyl-4-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-[2-(dimethylamino)ethyl]-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-oxopyrrolidine-3-carboxamide
(3S,9aR)-8-(cyclohexylmethyl)-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-cyclopentyl-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
3-{[1-(4-chloro-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]methyl}benzamide
8-[(6-chloropyridin-2-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[3-(4-fluorophenoxy)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
N-butyl-2-{1-[4-hydroxy-2-(4-methylphenyl)pyrimidin-5-yl]-N-methylformamido}acetamide
4-{2-[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]propyl}phenol
2-methyl-2-(2-{[(3-methylpyridin-2-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
2-cyclopropyl-9-[(4-methoxy-2,3-dimethylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(8-methoxyquinolin-2-yl)-3,9-diazaspiro[5.6]dodecan-10-one
4,4-difluoro-1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidine
3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
[2-(4-butylphenyl)pyridin-4-yl]methanol