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[(3R,5R)-5-[(dimethylamino)methyl]-1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-3-yl]methanol
5-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
2,3,6-trifluoro-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}benzamide
ethyl 3-({1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)hexanoate
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-2-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}pyrimidine
1-(2-cyclohexylethyl)-3-hydroxy-3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)piperidin-2-one
1-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-3-(1-methyl-1H-1,2,3-benzotriazol-5-yl)urea
(4aS,8aR)-N-benzyl-4a-(hydroxymethyl)-N-methyl-decahydro-1,6-naphthyridine-6-sulfonamide
6-(2-methoxyphenyl)-N-methylpyridine-2-carboxamide
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[2-(propan-2-yl)pyrimidine-4-carbonyl]-1,4-diazepane
3-methyl-1-[(4-methylphenyl)methyl]-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazin-2-one
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
2-oxo-2-[4-oxo-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-N-phenylacetamide
N-{2-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylmethanesulfonamide
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[4-(thian-4-yl)piperazin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
2-{[1-(4-chloro-1H-pyrrole-2-carbonyl)piperidin-4-yl]oxy}pyrimidine
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(pyridin-2-yl)acetamide
methyl 5-cyano-2-methyl-6-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]pyridine-3-carboxylate
[1-(1,3-benzothiazole-6-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
methyl 2-(diethylsulfamoyl)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-cyclobutyl-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-ethyl-1H-pyrazole-5-carboxamide
1-cyclohexyl-3-(cyclopropylmethyl)-5-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-3-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}-3-[2-(pyrrolidin-1-yl)ethyl]urea
1-benzyl-3-cyclopropyl-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazole
(4aS,7aR)-1-[(3,4-dimethylphenyl)methyl]-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[4-(1,3,7-trimethyl-1H-indole-2-carbonyl)-1,4-oxazepan-6-yl]methanol
(1S,2R)-N1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-N2-(prop-2-en-1-yl)cyclohexane-1,2-dicarboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[4-(2-hydroxyethoxy)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]acetamide
N'-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)butanediamide
3-methyl-5-(1-{2-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}propyl)-1,2,4-oxadiazole
1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
4-{[(3-methylthiophen-2-yl)methyl]amino}-N-(pyridin-4-ylmethyl)benzamide
N-[2-(4-hydroxyphenyl)ethyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-5-methoxybenzamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
[(3R,4R)-1-(6-cyclopropylpyrimidin-4-yl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-benzyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}pyrrolidin-3-amine
(4aS,8aR)-6-[2-(2-fluorophenyl)acetyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-(morpholin-4-yl)-3-{1-[(3-phenoxyphenyl)methyl]piperidin-4-yl}propan-1-one
N-[3-(4-{[2-(cyclohex-1-en-1-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-methylthiophene-2-carboxamide
1-{4-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
1-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carbonyl}cyclopropane-1-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]benzamide
3-{[(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)carbamoyl]methyl}-1,2,3-oxadiazol-3-ium-5-olate
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]cyclopropan-1-amine
(2R)-2-amino-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-phenylpropan-1-one