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(3S)-3-benzyl-4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-2-one
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(morpholine-4-carbonyl)benzene-1-sulfonamide
N-(2,3-dihydro-1H-inden-2-yl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(pyridin-3-yl)ethane-1,2-dione
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
methyl 5-({2-[2-(pyridin-3-yl)piperidin-1-yl]acetamido}methyl)furan-2-carboxylate
4,6-dimethyl-13-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
6-{1-[(6-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
5-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-(furan-2-ylmethyl)-N-methyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 4-[(3-methoxyphenyl)methyl]-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxylate
3-{2-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
9-ethyl-1-methyl-4-(pyridine-3-sulfonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2,6-diamino-4-[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(2S,4S)-4-amino-N,N-diethyl-1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-2-carboxamide
7-(2-methoxyquinoline-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
[(3R,5R)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
8-(4-aminopyrimidin-2-yl)-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
7-[2-(azepan-1-yl)acetyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3S,5R)-5-[(4-fluorophenyl)carbamoyl]-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)piperidine-3-carboxylic acid
[(5-ethylpyridin-2-yl)methyl](methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
(3S,4R)-1-[4-(1H-imidazol-1-yl)butanoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
4-[1-(4-chlorophenyl)cyclobutanecarbonyl]piperazine-1-sulfonamide
ethyl 4-[6-(2,1,3-benzothiadiazol-5-ylmethyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
N-(5-fluoro-2-methylphenyl)-2-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}propanamide
[2,2-dimethyl-3-(morpholin-4-yl)propyl][(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
[4-({[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl](methyl)amino}methyl)oxan-4-yl]methanol
1-methyl-N-{3-[methyl(phenyl)amino]propyl}-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}azepan-4-ol
3-(oxolan-3-yl)-5-[2-(pyrrolidin-1-yl)propan-2-yl]-1,2,4-oxadiazole
2-[2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamido]-2-methylpropanoic acid
2-[1-methyl-4-(naphthalen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
5-(2-chlorophenyl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]furan-2-carboxamide
3-[2-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
N-(1-cycloheptylpiperidin-3-yl)-2,6-difluorobenzamide
1-[2-({2-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-imidazol-1-yl}methyl)morpholin-4-yl]ethan-1-one
(4aS,8aR)-1-(3-hydroxypropyl)-6-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
5-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}-2-(pyridin-3-yl)pyrimidine
2-(4-{4-[ethyl(methyl)amino]pyrimidin-2-yl}-1H-pyrazol-1-yl)-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-(4-fluoro-3-methylphenyl)ethan-1-one
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
2-({[(3R,4R)-1-{[5-(2-fluorophenyl)furan-2-yl]methyl}-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-[5-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)furan-2-yl]benzonitrile
2-{3-[(3-fluorophenyl)amino]piperidine-1-carbonyl}-6-methylphenol
[1-(2H-1,3-benzodioxol-4-ylmethyl)-4-[(4-chlorophenyl)methyl]piperidin-4-yl]methanol
1-methyl-2-phenyl-4-{[1-(propan-2-yl)piperidin-4-yl]methyl}piperazine
3-chloro-5-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
8-methoxy-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1H-pyrazol-3-yl)phenol
2-phenyl-1-{1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-3-yl}ethan-1-one