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N-(2-{4-[1-(2,3-dimethylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)acetamide
8-(2-ethoxyacetyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N,2-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]thieno[2,3-d]pyrimidin-4-amine
[(1S,3S,3aS,6aR)-5-benzyl-3-(1-methyl-1H-imidazol-5-yl)-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-5-methylpiperidin-2-one
4-[4-(piperidine-1-carbonyl)phenoxy]-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
N-{[(2S,4S)-4-fluoro-1-(3-phenoxypropanoyl)pyrrolidin-2-yl]methyl}cyclopentanecarboxamide
N-(1H-indol-5-ylmethyl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
5-(4-cyclohexylphenyl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1,2,4-triazin-3-amine
3-ethyl-8-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(1-methyl-1H-pyrrol-2-yl)-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethane-1,2-dione
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
3-(4-chloro-1H-pyrazol-1-yl)-1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]propan-1-one
4-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}morpholine
2-(2H-1,2,3-benzotriazol-2-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]acetamide
N-(isoquinolin-5-ylmethyl)-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
4-{imidazo[1,2-a]pyridine-2-carbonyl}-1-methylpiperazin-2-one
1-[3-(2-methylphenoxy)azetidin-1-yl]-2-(pyrrolidin-1-yl)butan-1-one
(1R,2S,6R,7S)-4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-azatricyclo[5.2.2.02,6]undecane
N-[(4-acetamidophenyl)methyl]-2-{[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}acetamide
N-{[6,7-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-2,3-dimethyl-1H-indole-7-carboxamide
1-(dimethyl-1,3-thiazol-2-yl)-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-6-ol
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(oxan-4-yl)pyridin-2-amine
3-(4-hydroxyphenyl)-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-1H-pyrazole-5-carboxamide
N-{3-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-oxopropyl}acetamide
1-methyl-9-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
1-cyclopentyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]piperidine-3-carboxamide
3-(4-chloro-2-ethylphenyl)-1-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}urea
1-ethyl-3-(morpholine-4-carbonyl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-5-methyl-4,5,6,7-tetrahydro-2H-indazole
2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-6-methylpyridine-3-carbonitrile
1-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]-1,4-diazepane-6-carboxylic acid
3-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-chloro-2-methylphenyl)urea
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-(2-hydroxyethyl)-8-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-[4-(cyclopentylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
4-phenyl-N-{1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
methyl 3-methoxy-5-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}benzoate
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopropanesulfonamide
5-[1-(3-methylpyridin-2-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-2-(pyridin-2-yl)pyrimidine
1-methyl-3-phenyl-8-(9H-purin-6-yl)-1,8-diazaspiro[4.5]decan-2-one
3-[2-(1H-indol-3-yl)acetamido]-N-(2-methylphenyl)propanamide
6-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}quinoxaline
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-2-yl)propan-1-one
N3-tert-butyl-4-oxo-1-(propan-2-yl)-N5-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N'-(2-fluoro-5-methylphenyl)butanediamide
2-hydroxy-1-[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-methylpropan-1-one
N4-{[1-(methoxymethyl)cyclopropyl]methyl}-6-(propan-2-yl)pyrimidine-2,4-diamine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol