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4-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1,5-dimethyl-1H-pyrazole
2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
8-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}quinoline
2-[4-(cyclopent-3-ene-1-carbonyl)-6-hydroxy-1,4-diazepan-1-yl]pyridine-3-carboxamide
(4aS,7aR)-1-(4-methyl-1,3-thiazole-5-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-N-(piperidin-4-yl)pyridin-2-amine
N-methyl-4-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)benzene-1-sulfonamide
[1-ethyl-5-(5-phenyl-1,2-oxazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
1-[2-(2-butyl-4-methyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1,2-dihydroquinolin-2-one
N-(4-fluoro-2-methylphenyl)-3-[1-(2-phenylacetyl)piperidin-3-yl]propanamide
1-[4-(pyridin-2-yl)piperazin-1-yl]-3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]propan-1-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]piperazine
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-4-(piperidin-3-yl)benzamide
N-[2-(dimethylamino)ethyl]-1-[1-(3-phenylbutyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
N-methyl-3-(morpholine-4-carbonyl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[3-(1H-indol-1-yl)propyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
3-[5-(propan-2-yl)pyrimidin-4-yl]-3,9-diazaspiro[5.5]undecane
N-[(3S)-2-oxoazepan-3-yl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
2-amino-N-(furan-2-ylmethyl)-N-methyl-1,3-benzothiazole-5-carboxamide
4-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}pyridazine
2-[(cyclopropylmethyl)sulfanyl]-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
(1S,5R)-6-benzyl-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-acetyl-N-[1-(3-methylpyridin-2-yl)propyl]piperidine-4-carboxamide
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-3-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]propanamide
7-(3-chlorophenyl)-4-(2-ethyl-6-methylpyrimidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1S,4R)-2-[(2,6-dichlorophenyl)methyl]-2-azabicyclo[2.2.1]heptan-3-one
N-[3-(2-methoxyphenoxy)propyl]-N-methyl-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-[(4-methoxy-3-methylphenyl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
N-(oxolan-2-ylmethyl)-5-[(4-phenyl-1,4-diazepan-1-yl)methyl]pyrimidin-2-amine
N-ethyl-5-{1-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
8-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-2,1,3-benzothiadiazole
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
(2R,3R)-3-{[2-(pyridin-2-ylsulfanyl)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-[(2S)-2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-1-(propan-2-yl)piperidine
2-fluoro-4-methyl-N-{2-[4-(propan-2-yl)morpholin-2-yl]ethyl}benzene-1-sulfonamide
7-(1,3-benzothiazol-2-yl)-4-(oxolane-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2,8-dimethylquinoline-4-carboxamide
N-[2-(2-ethoxyphenyl)ethyl]-2-fluoro-5-sulfamoylbenzamide
2-[(4aR,7aS)-4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
6-[(3-fluorophenyl)methoxy]-4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1-(2-methylpropyl)-1,4-diazepan-2-one
2-[8-(butan-2-yl)-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
2-(dimethylamino)-N-methyl-N-{[1-(2-methylphenyl)-1H-1,2,3,4-tetrazol-5-yl](phenyl)methyl}acetamide
[(2-ethoxyphenyl)methyl](ethyl)[(3-methyl-1H-pyrazol-5-yl)methyl]amine
4-[(cyclopropylmethyl)sulfamoyl]-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
(1S,5R)-3-[(3-ethoxyphenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-({3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-4-methoxyphenol
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-3-methoxypropanamide
5-butyl-1'-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4,4-difluoropiperidine