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1-(4-fluoro-3-methoxyphenyl)-2-(furan-2-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
(3aR,6aR)-2-cyclopentyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
1-[(3-chlorophenyl)methyl]-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(propan-2-yl)pyrimidine-4-carboxamide
N-[2-(4-fluorophenyl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(dimethylamino)-N-[2-methyl-5-({[(5-methylpyrazin-2-yl)methyl]carbamoyl}amino)phenyl]acetamide
methyl 5-({[3-(2-hydroxyethoxy)phenyl]methyl}amino)-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-(2-amino-4-methyl-6-{methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]amino}pyrimidin-5-yl)propanoic acid
1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-{[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]sulfonyl}benzoic acid
2-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-8-methoxyquinoline
2-[2-(3-ethyl-3-hydroxypiperidin-1-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
1-methyl-N-[3-(methylsulfanyl)propyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(4-fluorophenyl)methyl]-2-methanesulfonyl-N-(oxolan-2-ylmethyl)acetamide
1-(4-methoxyphenyl)-2,2-dimethyl-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazine
4-[(1-propylpiperidin-4-yl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
5-[6-(thiomorpholin-4-yl)pyridazin-3-yl]isoquinoline
2-cyclopropanecarbonyl-8-[(3-fluoro-2-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
ethyl 1-[3-(1,2-oxazolidin-2-yl)propanoyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-2-(5-methyl-1H-pyrazol-1-yl)acetamide
N-[1-(4-methylphenyl)ethyl]-2-{[(3-methylthiophen-2-yl)methyl]amino}acetamide
2-[1-(2-methoxyethyl)-2,5-dimethyl-1H-pyrrol-3-yl]-1-methyl-1H-1,3-benzodiazole
methyl({[1-(morpholin-4-yl)cyclohexyl]methyl})(1H-pyrazol-3-ylmethyl)amine
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[4-(morpholin-4-yl)butyl]amine
7-methyl-3-({methyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-methoxy-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]pyridine-3-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]benzamide
5,6-dimethyl-2-[3-(morpholin-4-ylmethyl)phenyl]pyridine-3-carboxamide
2-{4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepan-1-yl}-N-ethylpyridine-3-carboxamide
1-[(2-phenyl-1,3-thiazol-5-yl)methyl]-4-(1,3-thiazol-2-yl)piperazine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(1H-pyrrol-1-yl)pentanamide
(1R,5S)-3-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
({4-[1-(5-chloropyridine-3-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
1-[3-({2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)phenyl]imidazolidin-2-one
3-methyl-7-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[4-(pyridin-3-yloxy)phenyl]-1-(1,3-thiazol-5-ylmethyl)piperidine-2-carboxamide
(3S,4R)-4-(2-methylphenyl)-1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidine-3-carboxylic acid
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(methylamino)ethan-1-one
8-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
3-{1-[(5-ethylthiophen-2-yl)sulfonyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
N-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-2-(trifluoromethyl)pyrimidin-4-amine
N-[1-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)piperidin-4-yl]acetamide
(1S,5R)-6-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
2-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-(thiophen-2-ylmethyl)acetamide